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Synthetic analogs of luteinizing hormone releasing hormone (LH-RH) substituted in position 6 and 10.

作者信息

Fujino M, Fukuda T, Shinagawa S, Kobayashi S, Yamazaki I

出版信息

Biochem Biophys Res Commun. 1974 Sep 9;60(1):406-13. doi: 10.1016/0006-291x(74)90219-8.

DOI:10.1016/0006-291x(74)90219-8
PMID:4608231
Abstract
摘要

相似文献

1
Synthetic analogs of luteinizing hormone releasing hormone (LH-RH) substituted in position 6 and 10.在第6位和第10位被取代的促黄体生成素释放激素（LH-RH）的合成类似物。
Biochem Biophys Res Commun. 1974 Sep 9;60(1):406-13. doi: 10.1016/0006-291x(74)90219-8.
2
Some analogs of luteinizing hormone releasing hormone (LH-RH) having intense ovulation-inducing activity.
Biochem Biophys Res Commun. 1974 Apr 23;57(4):1248-56. doi: 10.1016/0006-291x(74)90830-4.
3
Synthesis and biological activities of analogs of the luteinizing hormone-releasing hormone (LH-RH) modified in position 2.在第2位进行修饰的促黄体生成激素释放激素（LH-RH）类似物的合成及生物活性
J Med Chem. 1974 Sep;17(9):1016-9. doi: 10.1021/jm00255a025.
4
Further studies on the structure-activity relationships in the C-terminal part of luteinizing hormone-releasing hormone.
J Med Chem. 1973 Oct;16(10):1144-7. doi: 10.1021/jm00268a017.
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Presence of proline in position 3 for potent inhibition of the activity of the luteinizing hormone releasing hormone and of ovulation.脯氨酸位于第3位可有效抑制促黄体生成素释放激素的活性及排卵。
Biochem Biophys Res Commun. 1976 Oct 4;72(3):939-44. doi: 10.1016/s0006-291x(76)80222-7.
6
Synthesis and biological properties of (Leu-6)-LH-RH and (D-Leu-6,desGly-NH210)-LH-RH ethylamide.
Biochem Biophys Res Commun. 1974 Aug 19;59(4):1226-32. doi: 10.1016/0006-291x(74)90445-8.
7
Synthetic luteinizing hormone releasing factor. Short chain analogs.
J Med Chem. 1974 Feb;17(2):230-3. doi: 10.1021/jm00248a019.
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Synthesis and biological activities of analogs of luteinizing hormone releasing hormone (LH-RH).促黄体生成素释放激素（LH-RH）类似物的合成及生物活性
Biochem Biophys Res Commun. 1972 Nov 1;49(3):698-705. doi: 10.1016/0006-291x(72)90467-6.
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Analogs of luteinizing hormone releasing factor (LRF). Synthesis and biological activity of ((Nalpha-Me)Leu-7)LRF and (D-Ala-6,(Nalpha-Me)Leu-7)LRF.促黄体生成素释放因子（LRF）类似物。（（Nα-甲基）亮氨酸-7）LRF和（D-丙氨酸-6，（Nα-甲基）亮氨酸-7）LRF的合成及生物活性
Biochem Biophys Res Commun. 1975 Apr 7;63(3):801-6. doi: 10.1016/s0006-291x(75)80454-2.
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Inhibitory analogues of the luteinizing hormone-releasing hormone having D-aromatic residues in positions 2 and 6 and variation in position 3.在第2位和第6位具有D-芳香族残基且第3位有变异的促黄体生成激素释放激素抑制类似物。
J Med Chem. 1978 Jan;21(1):120-3. doi: 10.1021/jm00199a024.

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