(1-beta-mercapto-beta,beta-diethylpropionic acid,4-leucine)-8-lysine-vasopressin and (1-beta-mercapto-beta,beta-diethylpropionic acid,4-leucine)oxytocin, compounds possessing antihormonal properties.
作者信息
Dyckes D F, Nestor J J, Ferger M F, Du Vigneaud V, Chan W Y
出版信息
J Med Chem. 1974 Sep;17(9):969-72. doi: 10.1021/jm00255a012.
PMID:4855467
Abstract
摘要
相似文献
1
(1-beta-mercapto-beta,beta-diethylpropionic acid,4-leucine)-8-lysine-vasopressin and (1-beta-mercapto-beta,beta-diethylpropionic acid,4-leucine)oxytocin, compounds possessing antihormonal properties.（1-β-巯基-β，β-二乙基丙酸，4-亮氨酸）-8-赖氨酸-加压素和（1-β-巯基-β，β-二乙基丙酸，4-亮氨酸）催产素，具有抗激素特性的化合物。
J Med Chem. 1974 Sep;17(9):969-72. doi: 10.1021/jm00255a012.
2
(1-Beta-mercapto-beta,beta-diethylpropionic acid)-8-lysine-vasopressin, a potent inhibitor of 8-lysine-vasopressin and of oxytocin.（1-巯基-β，β-二乙基丙酸）-8-赖氨酸-加压素，一种8-赖氨酸-加压素和催产素的强效抑制剂。
J Med Chem. 1974 Feb;17(2):250-2. doi: 10.1021/jm00248a028.
3
Synthesis and some of the pharmacological properties of (4-leucine)-8-lysine-vasopressin and (1-deamino,4-leucine)-8-lysine-vasopressin.（4-亮氨酸）-8-赖氨酸加压素和（1-去氨基，4-亮氨酸）-8-赖氨酸加压素的合成及其某些药理特性
J Med Chem. 1973 Jul;16(7):843-7. doi: 10.1021/jm00265a022.
4
[1-Beta-mercapto-beta,beta-pentamethylenepropionic acid]oxytocin, a potent inhibitor of oxytocin.[1-巯基-β,β-五亚甲基丙酸]催产素，一种强效催产素抑制剂。
J Med Chem. 1975 Mar;18(3):284-7. doi: 10.1021/jm00237a015.
5
Study of pituitary hormone analogs for their inhibitory properties and resistance to carboxamidopeptidases: (9-L-proline)oxytocin, (9-L-glutamic acid)oxytocin, and (8-L-lysine,9-glycine methylamide)oxytocin.垂体激素类似物的抑制特性及其对羧肽酶抗性的研究：（9-L-脯氨酸）催产素、（9-L-谷氨酸）催产素和（8-L-赖氨酸，9-甘氨酸甲酰胺）催产素。
J Med Chem. 1974 Dec;17(12):1294-8. doi: 10.1021/jm00258a013.
6
Synthesis and some pharmacological properties of [1-beta-mercapto-beta,beta-diethylpropionic acid,2-(3,5-dibromo-L-tyrosine)]oxytocin.
J Med Chem. 1975 Dec;18(12):1262-4. doi: 10.1021/jm00246a021.
7
Synthesis and certain pharmacological properties of lysine-vasopressinoic acid methylamide and lysine-vasopressinoic acid dimethylamide.赖氨酸 - 加压素酸甲酰胺和赖氨酸 - 加压素酸二甲酰胺的合成及某些药理学性质
J Med Chem. 1972 May;15(5):486-8. doi: 10.1021/jm00275a012.
8
Synthetic antagonists of in vivo responses by the rat uterus to oxytocin.大鼠子宫对催产素体内反应的合成拮抗剂。
J Med Chem. 1979 May;22(5):565-9. doi: 10.1021/jm00191a019.
9
Synthesis of three oxytocin analogs related to (1-deaminopenicillamine)oxytocin possessing antioxytocic acitvity.
J Med Chem. 1972 Feb;15(2):123-6. doi: 10.1021/jm00272a001.
10
Solid phase synthesis of (3,4-dileucine)-oxytocin and a study of some of its pharmacological properties.（3,4-二亮氨酸）-催产素的固相合成及其部分药理性质研究
J Med Chem. 1972 Jan;15(1):11-2. doi: 10.1021/jm00271a004.
引用本文的文献
1
Relative conformational rigidity in oxytocin and (1-penicillamine)-oxytocin: a proposal for the relationship of conformational flexibility to peptide hormone agonism and antagonism.催产素和（1-青霉胺）-催产素中的相对构象刚性：关于构象灵活性与肽类激素激动作用和拮抗作用关系的一项提议。
Proc Natl Acad Sci U S A. 1977 Apr;74(4):1373-7. doi: 10.1073/pnas.74.4.1373.
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