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Quantitative structure-activity relationships of antineoplastic drugs: nitrosoureas and triazenoimidazoles.

作者信息

Hansch C, Smith N, Engle R, Wood H

出版信息

Cancer Chemother Rep. 1972 Aug;56(4):443-56.

PMID:5081587
Abstract
摘要

相似文献

1
Quantitative structure-activity relationships of antineoplastic drugs: nitrosoureas and triazenoimidazoles.
Cancer Chemother Rep. 1972 Aug;56(4):443-56.
2
Value of cytosine arabinoside (NSC-63878) plus 5-(3,3-dimethyl-1-triazeno)imidazole-4-carboxamide (NSC-45388) therapy in advanced murine L1210 leukemia and enhancement of the combination with sequential doses of methotrexate (NSC-740) or 1,3-bis(2-chloroethyl)-1-nitrosourea (BCNU; NSC-409962).阿糖胞苷（NSC - 63878）加5 -（3,3 - 二甲基 - 1 - 三氮烯）咪唑 - 4 - 甲酰胺（NSC - 45388）疗法在晚期小鼠L1210白血病中的价值以及与甲氨蝶呤（NSC - 740）或1,3 - 双（2 - 氯乙基）-1 - 亚硝基脲（卡莫司汀；NSC - 409962）序贯剂量联合使用时疗效的增强。
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Recent advances in the biochemical pharmacology of selected alkylating agents.某些烷化剂的生化药理学最新进展。
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Therapy of malignant melanoma with an imidazole carboxamide and bis-chloroethyl nitrosourea.用咪唑甲酰胺和双氯乙基亚硝脲治疗恶性黑色素瘤。
Cancer. 1972 Dec;30(6):1457-61. doi: 10.1002/1097-0142(197212)30:6<1457::aid-cncr2820300607>3.0.co;2-5.
5
Comparative studies on the chemical stability and therapeutic effectiveness of water-insoluble 5-(3,3-bis(2-chloroethyl)-1-triazeno)imidazole-4-carboxamide (NSC-82196) and its water-soluble hydrochloride against L1210 mouse leukemia.
Cancer Chemother Rep. 1973 Nov-Dec;57(4):383-91.
6
Evaluation of antileukemic agents in advanced leukemia L1210 in mice. X.小鼠晚期白血病L1210中抗白血病药物的评价。X。
Cancer Chemother Rep 2. 1972 Nov;3(1):1-69.
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Contributions of nitrosoureas to cancer treatment.亚硝基脲类药物在癌症治疗中的作用。
Cancer Treat Rep. 1986 Jan;70(1):31-41.
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Relationship of structure to anticancer activity and toxicity of the nitrosoureas in animal systems.动物系统中亚硝基脲类的结构与抗癌活性及毒性的关系。
Cancer Treat Rep. 1986 Jan;70(1):13-30.
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Combination therapy: some concepts and results.
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Antitumor structure-activity relations. Nitrosoureas vs. L-1210 leukemia.抗肿瘤构效关系。亚硝基脲类与L - 1210白血病
J Med Chem. 1980 Oct;23(10):1095-101. doi: 10.1021/jm00184a007.

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