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Specificity of porcine pancreatic elastase, human leukocyte elastase and cathepsin G. Inhibition with peptide chloromethyl ketones.

作者信息

Powers J C, Gupton B F, Harley A D, Nishino N, Whitley R J

出版信息

Biochim Biophys Acta. 1977 Nov 23;485(1):156-66. doi: 10.1016/0005-2744(77)90203-0.

DOI:10.1016/0005-2744(77)90203-0
PMID:562189
Abstract
摘要

相似文献

1
Specificity of porcine pancreatic elastase, human leukocyte elastase and cathepsin G. Inhibition with peptide chloromethyl ketones.猪胰弹性蛋白酶、人白细胞弹性蛋白酶和组织蛋白酶G的特异性。肽氯甲基酮对其的抑制作用。
Biochim Biophys Acta. 1977 Nov 23;485(1):156-66. doi: 10.1016/0005-2744(77)90203-0.
2
Specificity and reactivity of human leukocyte elastase, porcine pancreatic elastase, human granulocyte cathepsin G, and bovine pancreatic chymotrypsin with arylsulfonyl fluorides. Discovery of a new series of potent and specific irreversible elastase inhibitors.人白细胞弹性蛋白酶、猪胰弹性蛋白酶、人粒细胞组织蛋白酶G以及牛胰凝乳蛋白酶与芳基磺酰氟的特异性和反应活性。新型强效且特异性不可逆弹性蛋白酶抑制剂系列的发现。
J Biol Chem. 1982 May 10;257(9):5077-84.
3
Amino acids and peptides. XXX. Synthesis of eglin c (41-49) and eglin c (60-63) and examination of their inhibitory activity towards human leukocyte elastase, cathepsin G, porcine pancreatic elastase and alpha-chymotrypsin.氨基酸与肽。XXX。埃格林c(41 - 49)和埃格林c(60 - 63)的合成及其对人白细胞弹性蛋白酶、组织蛋白酶G、猪胰弹性蛋白酶和α-胰凝乳蛋白酶抑制活性的检测。
Chem Pharm Bull (Tokyo). 1991 Jan;39(1):184-6. doi: 10.1248/cpb.39.184.
4
Unusual reactivity of trifluoroacetyl peptide chloromethyl ketones with pancreatic elastase.三氟乙酰肽氯甲基酮与胰腺弹性蛋白酶的异常反应性。
J Am Chem Soc. 1978 Feb 1;100(3):1005-7. doi: 10.1021/ja00471a076.
5
Similarities between human and rat leukocyte elastase and cathepsin G.人类与大鼠白细胞弹性蛋白酶和组织蛋白酶G之间的相似性。
Eur J Biochem. 1984 Oct 1;144(1):1-9. doi: 10.1111/j.1432-1033.1984.tb08423.x.
6
Studies on reactivity of human leukocyte elastase, cathepsin G, and porcine pancreatic elastase toward peptides including sequences related to the reactive site of alpha 1-protease inhibitor (alpha 1-antitrypsin).关于人白细胞弹性蛋白酶、组织蛋白酶G和猪胰弹性蛋白酶对包括与α1-蛋白酶抑制剂(α1-抗胰蛋白酶)反应位点相关序列的肽的反应性研究。
Biochemistry. 1980 Aug 19;19(17):3973-8. doi: 10.1021/bi00558a013.
7
Human leukocyte and porcine pancreatic elastase: X-ray crystal structures, mechanism, substrate specificity, and mechanism-based inhibitors.人白细胞弹性蛋白酶和猪胰弹性蛋白酶:X射线晶体结构、作用机制、底物特异性及基于机制的抑制剂
Biochemistry. 1989 Mar 7;28(5):1951-63. doi: 10.1021/bi00431a001.
8
A new class of heterocyclic serine protease inhibitors. Inhibition of human leukocyte elastase, porcine pancreatic elastase, cathepsin G, and bovine chymotrypsin A alpha with substituted benzoxazinones, quinazolines, and anthranilates.一类新型杂环丝氨酸蛋白酶抑制剂。用取代苯并恶嗪酮、喹唑啉和邻氨基苯甲酸酯对人白细胞弹性蛋白酶、猪胰弹性蛋白酶、组织蛋白酶G和牛胰凝乳蛋白酶Aα的抑制作用。
J Biol Chem. 1982 May 10;257(9):5085-91.
9
Active site mapping of the serine proteases human leukocyte elastase, cathepsin G, porcine pancreatic elastase, rat mast cell proteases I and II. Bovine chymotrypsin A alpha, and Staphylococcus aureus protease V-8 using tripeptide thiobenzyl ester substrates.使用三肽硫代苄酯底物对丝氨酸蛋白酶人白细胞弹性蛋白酶、组织蛋白酶G、猪胰弹性蛋白酶、大鼠肥大细胞蛋白酶I和II、牛胰凝乳蛋白酶Aα以及金黄色葡萄球菌蛋白酶V-8进行活性位点图谱分析。
Biochemistry. 1984 Jun 19;23(13):2995-3002. doi: 10.1021/bi00308a023.
10
Inhibition of the human leukocyte endopeptidases elastase and cathepsin G and of porcine pancreatic elastase by N-oleoyl derivatives of heparin.肝素的N-油酰基衍生物对人白细胞内肽酶弹性蛋白酶和组织蛋白酶G以及猪胰弹性蛋白酶的抑制作用。
Biochem Pharmacol. 1993 Nov 2;46(9):1545-9. doi: 10.1016/0006-2952(93)90321-m.

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