Kinetic parameters of narcotic agonists and antagonists, with particular reference to N-allylnoroxymorphone (naloxone).
作者信息
Kosterlitz H W, Watt A J
出版信息
Br J Pharmacol Chemother. 1968 Jun;33(2):266-76. doi: 10.1111/j.1476-5381.1968.tb00988.x.
Abstract
摘要
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STUDIES ON THE HUMAN ADDICTION LIABILITY OF 2'-HYDROXY-5-9-DIMETHYL-2-(3,3-DIMETHYLALLYL)-6,7-BENZOMORPHAN (WIN 20,228): A WEAK NARCOTIC ANTAGONIST.
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N-Allylnoroxy-morphone: a new potent narcotic antagonist.
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Studies of analgesic drugs. VII. Morphine antagonists as analgesics.
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[Relationship between the effects of analgesics and sympathomimetics on guinea pig small intestines].
Naunyn Schmiedebergs Arch Exp Pathol Pharmakol. 1958;233(1):112-24.
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Synthetic substances with morphine-like effect: clinical experience; potency, side-effects, addiction liability.
Bull World Health Organ. 1957;17(4-5):569-863.
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A modification of receptor theory.
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8
The human pharmacology and abuse potential of N-allylnoroxymorphone (naloxone).
J Pharmacol Exp Ther. 1967 Aug;157(2):420-6.
9
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Br J Pharmacol Chemother. 1966 Sep;27(3):514-27. doi: 10.1111/j.1476-5381.1966.tb01864.x.
10
Drug interaction in the field of analgesic drugs.
Proc R Soc Med. 1965 Nov;58(11 Part 2):978-83. doi: 10.1177/003591576505811P207.
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