Morphine analgesia after intrathecal administration of a narcotic agonist, chloroxymorphamine and antagonist, chlornaltrexamine.
作者信息
Larson A A, Armstrong M J
出版信息
Eur J Pharmacol. 1980 Nov 7;68(1):25-31. doi: 10.1016/0014-2999(80)90056-4.
PMID:6161013
Abstract
摘要
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1
Morphine analgesia after intrathecal administration of a narcotic agonist, chloroxymorphamine and antagonist, chlornaltrexamine.鞘内注射麻醉性激动剂氯羟吗啡和拮抗剂氯纳曲胺后的吗啡镇痛作用。
Eur J Pharmacol. 1980 Nov 7;68(1):25-31. doi: 10.1016/0014-2999(80)90056-4.
2
Pharmacological studies with an alkylating narcotic agonist, chloroxymorphamine, and antagonist, chlornaltrexamine.
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Chloroxymorphamine, and opioid receptor site-directed alkylating agent having narcotic agonist activity.氯氧吗啡，一种具有麻醉激动剂活性的阿片受体位点定向烷基化剂。
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4
Irreversible opiate agonists and antagonists. II. Evidence against a bivalent mechanism of action for opiate azines and diacylhydrazones.不可逆阿片类激动剂和拮抗剂。II. 反对阿片嗪和二酰基腙二价作用机制的证据。
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5
Antagonism by chlornaltrexamine of some effects of delta 9-tetrahydrocannabinol in rats.氯纳曲明对大鼠中δ9-四氢大麻酚某些作用的拮抗作用。
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6
Long-acting opiate agonists and antagonists: 14-hydroxydihydromorphinone hydrazones.
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7
Synthesis and pharmacologic characterization of an alkylating analogue (chlornaltrexamine) of naltrexone with ultralong-lasting narcotic antagonist properties.具有超长效麻醉拮抗特性的纳曲酮烷基化类似物（氯甲纳曲酮）的合成及药理学特性研究
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8
6beta-[N,N-Bis(2-chloroethyl)amino]-17-(cyclopropylmethyl)-4,5alpha-epoxy-3,14-dihydroxymorphinan(chlornaltrexamine) a potent opioid receptor alkylating agent with ultralong narcotic antagonist actitivty.6β-[N,N-双（2-氯乙基）氨基]-17-（环丙基甲基）-4,5α-环氧-3,14-二羟基吗啡喃（氯纳曲明），一种具有超长麻醉拮抗活性的强效阿片受体烷基化剂。
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9
Augmentation of spinal morphine analgesia and inhibition of tolerance by low doses of mu- and delta-opioid receptor antagonists.低剂量μ-和δ-阿片受体拮抗剂增强脊髓吗啡镇痛作用并抑制耐受性。
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Irreversible opiate agonists and antagonists. III. Phenylhydrazone derivatives of naloxone and oxymorphone.不可逆阿片类激动剂和拮抗剂。III. 纳洛酮和羟吗啡酮的苯腙衍生物。
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