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Structure-activity relationships of enkephalin-like peptides.

作者信息

Morley J S

出版信息

Annu Rev Pharmacol Toxicol. 1980;20:81-110. doi: 10.1146/annurev.pa.20.040180.000501.

DOI:10.1146/annurev.pa.20.040180.000501

PMID:6247963

Abstract

摘要

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Structure-activity relationships of enkephalin-like peptides.

Annu Rev Pharmacol Toxicol. 1980;20:81-110. doi: 10.1146/annurev.pa.20.040180.000501.

Effects of enkephalin in analogues on prolactin release in the rat.

Life Sci. 1978 Jun 5;22(21):1931-7. doi: 10.1016/0024-3205(78)90480-0.

Stimulation of growth hormone and prolactin release by a potent enkephalin analog.

FEBS Lett. 1978 Apr 15;88(2):208-10. doi: 10.1016/0014-5793(78)80175-6.

Potent prolactin and growth hormone releasing activity of more analogues of Met-enkephalin.

Nature. 1977 Aug 11;268(5620):544-7. doi: 10.1038/268544a0.

[Endogenous polypeptides with morphine-like activity (enkephalins, endorphins, anodynin) (a review of the literature)].

Farmakol Toksikol. 1978 Mar-Apr;41(2):245-56.

Potent analgesic activity of the enkephalin-like tetrapeptide H-Tyr-D-Ala-Gly-Phe-NH2.

Life Sci. 1978 Oct 2;23(13):1371-6. doi: 10.1016/0024-3205(78)90396-x.

[Enkephalins, endorphins (author's transl)].

J Pharm Belg. 1979 Jan-Feb;34(1):35-43.

Opioid activity of synthetic and naturally occurring enkephalin peptides.

Biochem Pharmacol. 1979 Nov 15;28(22):3333-7. doi: 10.1016/0006-2952(79)90129-1.

Interactions of leucine enkephalin and narcotics with opioid receptors.

Mol Pharmacol. 1981 Mar;19(2):236-41.

Effects of the synthetic enkephalin analogue FK 33-824 in man.

Nature. 1978 Apr 20;272(5655):729-30. doi: 10.1038/272729a0.

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Structure-activity relationships of enkephalin-like peptides.

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