Archer S, Osei-Gyimah P, Silbering S
J Med Chem. 1980 May;23(5):516-9. doi: 10.1021/jm00179a009.
A series of 4-[N-(aminoalkyl)amino]-1,2-dimethoxynaphthalenes was prepared and tested for radical curative activity in rhesus monkeys infected with P. cynomolgi. Some radical curative activity was observed.
制备了一系列4-[N-(氨基烷基)氨基]-1,2-二甲氧基萘,并在感染食蟹猴疟原虫的恒河猴中测试其根治活性。观察到了一些根治活性。