大鼠离体灌流心脏中儿茶酚-O-甲基转移酶抑制剂U-0521与托酚酮乙酰胺性质的比较研究 - Suppr

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超能文献

A comparative study of the properties of the catechol-O-methyltransferase inhibitors, U-0521 and tropolone acetamide, in rat perfused heart.

作者信息

Bryan L J, Fleig H, Trendelenburg U

出版信息

Naunyn Schmiedebergs Arch Pharmacol. 1983 Feb;322(1):6-19. doi: 10.1007/BF00649346.

DOI:10.1007/BF00649346

PMID:6843690

Abstract

摘要

相似文献

A comparative study of the properties of the catechol-O-methyltransferase inhibitors, U-0521 and tropolone acetamide, in rat perfused heart.大鼠离体灌流心脏中儿茶酚-O-甲基转移酶抑制剂U-0521与托酚酮乙酰胺性质的比较研究

Naunyn Schmiedebergs Arch Pharmacol. 1983 Feb;322(1):6-19. doi: 10.1007/BF00649346.

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Extraneuronal removal, accumulation and O-methylation of isoprenaline in the perfused heart.灌注心脏中异丙肾上腺素的非神经元性清除、蓄积及O-甲基化作用

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Comparative effect of tropolone and diosmin on venous COMT and sympathetic activity in rat.托酚酮和地奥司明对大鼠静脉儿茶酚-O-甲基转移酶和交感神经活性的比较作用。

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Possible activation of intracellular beta-adrenoceptors by extraneuronally accumulated isoprenaline in perfused rat heart.灌注大鼠心脏中细胞外积聚的异丙肾上腺素可能激活细胞内β-肾上腺素能受体。

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引用本文的文献

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Naunyn Schmiedebergs Arch Pharmacol. 1995 Apr;351(4):408-16. doi: 10.1007/BF00169082.

The isotope effect of tritium in 3H-noradrenaline.3H-去甲肾上腺素中氚的同位素效应。

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The extraneuronal compartments for the distribution of isoprenaline in the rat heart.大鼠心脏中异丙肾上腺素分布的神经外间隙。

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The influence of inhibition of catechol-O-methyl transferase or of monoamine oxidase on the extraneuronal metabolism of 3H-(-)-noradrenaline in the rat heart.儿茶酚-O-甲基转移酶抑制或单胺氧化酶抑制对大鼠心脏中3H-(-)-去甲肾上腺素细胞外代谢的影响。

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The kinetic characteristics of the extraneuronal Q-methylating system of the dog saphenous vein and the supersensitivity to catecholamines caused by its inhibition.犬隐静脉神经外Q-甲基化系统的动力学特性及其抑制所引起的对儿茶酚胺的超敏反应。

Naunyn Schmiedebergs Arch Pharmacol. 1984 Aug;327(1):48-55. doi: 10.1007/BF00504991.

Kinetic constants of isoprenaline and corticosterone for extraneuronal uptake in different cell types from various tissues.不同组织中不同细胞类型对异丙肾上腺素和皮质酮的非神经元摄取动力学常数。

Naunyn Schmiedebergs Arch Pharmacol. 1984 Jan;325(1):54-61. doi: 10.1007/BF00507054.

Saturation of monoamine oxidase by intraneuronal noradrenaline accumulation.神经元内去甲肾上腺素积累导致单胺氧化酶饱和。

Naunyn Schmiedebergs Arch Pharmacol. 1984 Dec;328(2):135-41. doi: 10.1007/BF00512062.

The outward transport of catecholamines mediated by uptake2 of the rat heart.大鼠心脏摄取2介导的儿茶酚胺外向转运。

Naunyn Schmiedebergs Arch Pharmacol. 1985 Sep;330(3):203-11. doi: 10.1007/BF00572435.

本文引用的文献

The uptake of catechol amines at high perfusion concentrations in the rat isolated heart: A novel catechol amine uptake process.大鼠离体心脏在高灌注浓度下对儿茶酚胺的摄取：一种新的儿茶酚胺摄取过程。

Br J Pharmacol Chemother. 1965 Aug;25(1):18-33. doi: 10.1111/j.1476-5381.1965.tb01753.x.

CATECHOL-OMETHYL TRANSFERASE INHIBITORS. IN VITRO INHIBITION OF THE ENZYME IN MOUSE-BRAIN EXTRACT.儿茶酚 - O - 甲基转移酶抑制剂。对小鼠脑提取物中该酶的体外抑制作用。

Acta Pharmacol Toxicol (Copenh). 1964;21:205-14. doi: 10.1111/j.1600-0773.1964.tb01785.x.

OCCUPANCY OF ADRENERGIC RECEPTORS AND INHIBITION OF CATECHOL O-METHYL TRANSFERASE BY TROPOLONES.托酚酮对肾上腺素能受体的占据及儿茶酚-O-甲基转移酶的抑制作用

J Med Chem. 1963 Nov;6:755-9. doi: 10.1021/jm00342a028.

The effect of 4-methyltropolone on the metabolism of adrenaline.4-甲基托酚酮对肾上腺素代谢的影响。

Can J Biochem Physiol. 1963 Jul;41:1581-7.

Statistical estimations in enzyme kinetics.酶动力学中的统计估计

Biochem J. 1961 Aug;80(2):324-32. doi: 10.1042/bj0800324.

The determination of enzyme inhibitor constants.酶抑制剂常数的测定

Biochem J. 1953 Aug;55(1):170-1. doi: 10.1042/bj0550170.

Affinities of catecholamines for extraneuronal uptake in smooth muscle cells in trachealis muscle of guinea-pig.儿茶酚胺对豚鼠气管平滑肌细胞非神经元摄取的亲和力。

Naunyn Schmiedebergs Arch Pharmacol. 1980 Mar;311(2):139-46. doi: 10.1007/BF00510252.

A mathematical model representing the extraneuronal O-methylating system of the perfused rat heart.一种代表灌注大鼠心脏细胞外O-甲基化系统的数学模型。

Naunyn Schmiedebergs Arch Pharmacol. 1980 Feb;311(1):17-32. doi: 10.1007/BF00500298.

Kinetic analyses of the mechanisms of action of inhibitors of the extraneuronal uptake of adrenaline in smooth muscle cells of guinea-pig trachea.

Naunyn Schmiedebergs Arch Pharmacol. 1981 Jan;315(3):249-54. doi: 10.1007/BF00499842.

A kinetic analysis of the extraneuronal uptake and metabolism of catecholamines.儿茶酚胺的神经外摄取与代谢的动力学分析。

Rev Physiol Biochem Pharmacol. 1980;87:33-115. doi: 10.1007/BFb0030896.

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