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Multiple affinity states for noncompetitive blockers revealed by [3H]phencyclidine binding to acetylcholine receptor rich membrane fragments from Torpedo marmorata.

作者信息

Oswald R E, Heidmann T, Changeux J P

出版信息

Biochemistry. 1983 Jun 21;22(13):3128-36. doi: 10.1021/bi00282a015.

DOI:10.1021/bi00282a015
PMID:6882741
Abstract
摘要

相似文献

1
Multiple affinity states for noncompetitive blockers revealed by [3H]phencyclidine binding to acetylcholine receptor rich membrane fragments from Torpedo marmorata.
Biochemistry. 1983 Jun 21;22(13):3128-36. doi: 10.1021/bi00282a015.
2
Multiple sites of action for noncompetitive blockers on acetylcholine receptor rich membrane fragments from torpedo marmorata.非竞争性阻滞剂对电鳐富含乙酰胆碱受体的膜片段的多个作用位点。
Biochemistry. 1983 Jun 21;22(13):3112-27. doi: 10.1021/bi00282a014.
3
Demonstration and affinity labeling of a stereoselective binding site for a benzomorphan opiate on acetylcholine receptor-rich membranes from Torpedo electroplaque.
Proc Natl Acad Sci U S A. 1985 Feb;82(3):940-4. doi: 10.1073/pnas.82.3.940.
4
Multiple binding sites for phencyclidine on the nicotinic acetylcholine receptor from Torpedo ocellata electric organ.来自眼斑电鳐电器官的烟碱型乙酰胆碱受体上苯环己哌啶的多个结合位点。
Life Sci. 1984 Mar 12;34(11):1047-55. doi: 10.1016/0024-3205(84)90018-3.
5
Binding of phencyclidine to the detergent solubilized acetylcholine receptor from Torpedo marmorata.苯环利定与电鳐去污剂增溶的乙酰胆碱受体的结合。
Life Sci. 1983 Mar 7;32(10):1143-9. doi: 10.1016/0024-3205(83)90120-0.
6
Selective labeling of the delta subunit of the acetylcholine receptor by a covalent local anesthetic.通过共价局部麻醉剂对乙酰胆碱受体δ亚基进行选择性标记。
Biochemistry. 1981 Dec 8;20(25):7166-74. doi: 10.1021/bi00528a018.
7
Mechanism of phencyclidine binding to the acetylcholine receptor from Torpedo electroplaque.
Mol Pharmacol. 1984 May;25(3):360-8.
8
Allosteric properties of the acetylcholine receptor protein from Torpedo marmorata.电鳐乙酰胆碱受体蛋白的变构特性。
Cold Spring Harb Symp Quant Biol. 1983;48 Pt 1:35-52. doi: 10.1101/sqb.1983.048.01.006.
9
Effects of calcium on the binding of phencyclidine to acetylcholine receptor-rich membrane fragments from Torpedo californica electroplaque.
J Neurochem. 1983 Oct;41(4):1077-84. doi: 10.1111/j.1471-4159.1983.tb09054.x.
10
Desensitization of membrane-bound Torpedo acetylcholine receptor by amine noncompetitive antagonists and aliphatic alcohols: studies of [3H]acetylcholine binding and 22Na+ ion fluxes.胺类非竞争性拮抗剂和脂肪醇对膜结合型电鳐乙酰胆碱受体的脱敏作用：[3H]乙酰胆碱结合及22Na+离子通量的研究
Biochemistry. 1984 Aug 28;23(18):4023-33. doi: 10.1021/bi00313a003.

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Determinants of phencyclidine potency on the nicotinic acetylcholine receptors from muscle and electric organ.苯环利定对肌肉和电鳐电器官烟碱型乙酰胆碱受体作用强度的决定因素。
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Delimiting the binding site for quaternary ammonium lidocaine derivatives in the acetylcholine receptor channel.确定乙酰胆碱受体通道中季铵利多卡因衍生物的结合位点。
J Gen Physiol. 1998 Nov;112(5):611-21. doi: 10.1085/jgp.112.5.611.
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