Zalesov V S, Barteĭl B A, Fridman A L, Kolobov N A, Zalesov V V
Farmakol Toksikol. 1980 Mar-Apr;43(2):158-61.
It was established in experiments on mice and rats carried out according to conventional procedures that 13 adamantane derivatives have a greater tranquilizing activity than amantadine, 3-bromadamantoyl-1 diazomethane exerting a stronger effect than trioxazin. Two adamantane derivatives were found to have an anticonvulsant activity.
按照常规程序在小鼠和大鼠身上进行的实验表明,13种金刚烷衍生物比金刚烷胺具有更强的镇静活性,3-溴金刚烷甲酰基-1-重氮甲烷的效果比三恶嗪更强。发现两种金刚烷衍生物具有抗惊厥活性。