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用于抗菌和抗乙酰胆碱酯酶活性的取代4(3H)-喹唑啉酮衍生物的合成与评价。第3部分。

Synthesis and evaluation of substituted 4(3H)-quinazolone derivatives for antimicrobial and antiacetylcholinesterase activities. Part 3.

作者信息

Misra H K, Sen Gupta A K

出版信息

Pharmazie. 1982 Apr;37(4):254-6.

PMID:7100248
Abstract

The synthesis of some new 6,8-dibromo-2-N-(N-arylcarbamoyl) carbamoylmethylthio-3-aryl-4(3H)-quinazolone derivatives is described. The synthesized derivatives were screened for their antibacterial, antifungal and antiacetylcholinesterase activities in vitro. Most of the compounds exhibited interesting antimicrobial activities. The relation between this and their chemical structure has been studied.

摘要

描述了一些新型6,8 - 二溴 - 2 - N -（N - 芳基氨基甲酰基）氨基甲酰甲基硫代 - 3 - 芳基 - 4(3H)-喹唑啉酮衍生物的合成。对合成的衍生物进行了体外抗菌、抗真菌和抗乙酰胆碱酯酶活性筛选。大多数化合物表现出有趣的抗菌活性。并研究了其与化学结构之间的关系。

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