A new approach to conformationally restricted peptide analogs: rigid beta-bends. 1. Enkephalin as an example.

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作者信息

Krstenansky J L, Baranowski R L, Currie B L

出版信息

Biochem Biophys Res Commun. 1982 Dec 31;109(4):1368-74. doi: 10.1016/0006-291x(82)91928-3.

DOI:10.1016/0006-291x(82)91928-3

PMID:7168769

Abstract

摘要

相似文献

A new approach to conformationally restricted peptide analogs: rigid beta-bends. 1. Enkephalin as an example.

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Synthesis and biological activity of (D)Ala2,Leu5-enkephalins containing hydrophilic or hydrophobic moieties.含亲水或疏水基团的（D）丙氨酸2，亮氨酸5-脑啡肽的合成与生物活性

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Studies on peptides. CL. Syntheses of [D-His2]-analogs of enkephalin and adrenorphin and several [D-Arg2]enkephalin analogs.

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Bis-penicillamine enkephalins possess highly improved specificity toward delta opioid receptors.双青霉胺脑啡肽对δ阿片受体具有高度改善的特异性。

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[Differences in the action of enkephalins, beta-endorphin, and morphine on spontaneous rhythmic movements of the isolated rabbit ileum].

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