Tramadol hydrochloride--not just another opioid agonist.
作者信息
Eggers K, Power I
出版信息
Br J Clin Pharmacol. 1995 Mar;39(3):338-9. doi: 10.1111/j.1365-2125.1995.tb04460.x.
Abstract
摘要
相似文献
1
Tramadol hydrochloride--not just another opioid agonist.盐酸曲马多——并非普通的阿片类激动剂。
Br J Clin Pharmacol. 1995 Mar;39(3):338-9. doi: 10.1111/j.1365-2125.1995.tb04460.x.
2
Mechanistic and functional differentiation of tapentadol and tramadol.曲马多和酒石酸布托啡诺的作用机制和功能分化。
Expert Opin Pharmacother. 2012 Jul;13(10):1437-49. doi: 10.1517/14656566.2012.696097. Epub 2012 Jun 15.
3
Advances in perioperative pain management: use of medications with dual analgesic mechanisms, tramadol & tapentadol.围手术期疼痛管理的进展：使用具有双重镇痛机制的药物，曲马多和他喷他多。
Anesthesiol Clin. 2010 Dec;28(4):647-66. doi: 10.1016/j.anclin.2010.08.009.
4
The novel compound (+/-)-1-[10-((E)-3-Phenyl-allyl)-3,10-diaza-bicyclo[4.3.1]dec-3-yl]-propan-1-one (NS7051) attenuates nociceptive transmission in animal models of experimental pain; a pharmacological comparison with the combined mu-opioid receptor agonist and monoamine reuptake inhibitor tramadol.新型化合物（±）-1-[10-（（E）-3-苯基-烯丙基）-3,10-二氮杂双环[4.3.1]癸-3-基]-丙-1-酮（NS7051）可减轻实验性疼痛动物模型中的伤害性传递；与μ-阿片受体激动剂和单胺再摄取抑制剂曲马多联合用药的药理学比较。
Neuropharmacology. 2008 Feb;54(2):331-43. doi: 10.1016/j.neuropharm.2007.10.005. Epub 2007 Oct 16.
5
What is the main mechanism of tramadol?曲马多的主要作用机制是什么？
Naunyn Schmiedebergs Arch Pharmacol. 2015 Oct;388(10):999-1007. doi: 10.1007/s00210-015-1167-5. Epub 2015 Aug 21.
6
Tramadol antinociception is potentiated by clonidine through α₂-adrenergic and I₂-imidazoline but not by endothelin ET(A) receptors in mice.曲马朵的镇痛作用可被可乐定通过 α₂-肾上腺素能和 I₂-咪唑啉受体增强，但不能被内皮素 ET(A)受体增强，在小鼠中。
Eur J Pharmacol. 2012 May 15;683(1-3):109-15. doi: 10.1016/j.ejphar.2012.03.016. Epub 2012 Mar 16.
7
Tramadol enhances urethral continence function through µ-opioid receptors in rats.曲马多通过 μ 阿片受体增强大鼠尿道控尿功能。
Neurourol Urodyn. 2013 Jan;32(1):98-103. doi: 10.1002/nau.22274. Epub 2012 Jun 5.
8
Tramadol and strong opioid: synergistic or additive opioid effect?曲马多与强效阿片类药物：协同还是相加的阿片类效应？
Pain Pract. 2008 May-Jun;8(3):214-5; author reply 215-6. doi: 10.1111/j.1533-2500.2008.00193_1.x.
9
Tramadol hydrochloride: an overview of current use.盐酸曲马多：当前应用概述
Hosp Med. 1998 May;59(5):373-6.
10
Characterisation of tramadol, morphine and tapentadol in an acute pain model in Beagle dogs.在比格犬急性疼痛模型中对曲马多、吗啡和喷他佐辛的特性研究。
Vet Anaesth Analg. 2014 May;41(3):297-304. doi: 10.1111/vaa.12140. Epub 2014 Feb 27.
本文引用的文献
1
Complementary and synergistic antinociceptive interaction between the enantiomers of tramadol.曲马多对映体之间的互补性和协同性抗伤害感受相互作用。
J Pharmacol Exp Ther. 1993 Oct;267(1):331-40.
2
A comparison of the antinociceptive effects of imipramine, tramadol and anpirtoline.丙咪嗪、曲马多和安匹托林的抗伤害感受作用比较。
Br J Clin Pharmacol. 1994 Apr;37(4):325-33. doi: 10.1111/j.1365-2125.1994.tb04285.x.
3
Receptor binding, analgesic and antitussive potency of tramadol and other selected opioids.曲马多及其他选定阿片类药物的受体结合、镇痛及镇咳效力
Arzneimittelforschung. 1988 Jul;38(7):877-80.
4
Possible mechanisms of morphine analgesia.吗啡镇痛的可能机制。
Clin Neuropharmacol. 1991 Apr;14(2):131-47. doi: 10.1097/00002826-199104000-00003.
5
Tramadol: pain relief by an opioid without depression of respiration.曲马多：一种不抑制呼吸的阿片类镇痛药。
Anaesthesia. 1992 Apr;47(4):291-6. doi: 10.1111/j.1365-2044.1992.tb02166.x.
6
Opioid and nonopioid components independently contribute to the mechanism of action of tramadol, an 'atypical' opioid analgesic.阿片类和非阿片类成分独立地对曲马多（一种“非典型”阿片类镇痛药）的作用机制起作用。
J Pharmacol Exp Ther. 1992 Jan;260(1):275-85.
Zotero 插件