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Aspartyl alpha-((1-phenyl-3-(trifluoromethyl)-pyrazol-5-yl)oxy)methyl ketones as interleukin-1 beta converting enzyme inhibitors. Significance of the P1 and P3 amido nitrogens for enzyme-peptide inhibitor binding.

作者信息

Dolle R E, Singh J, Rinker J, Hoyer D, Prasad C V, Graybill T L, Salvino J M, Helaszek C T, Miller R E, Ator M A

机构信息

Department of Medicinal Chemistry, Sterling Winthrop Pharmaceuticals Research Division, Collegeville, Pennsylvania 19426.

出版信息

J Med Chem. 1994 Nov 11;37(23):3863-6. doi: 10.1021/jm00049a001.

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