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Transition state analysis and inhibitor design for enzymatic reactions.

作者信息

Schramm V L, Horenstein B A, Kline P C

机构信息

Department of Biochemistry, Albert Einstein College of Medicine, Bronx, New York 10461.

出版信息

J Biol Chem. 1994 Jul 15;269(28):18259-62.

PMID:8034566
Abstract
摘要

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Transition state analysis and inhibitor design for enzymatic reactions.酶促反应的过渡态分析与抑制剂设计
J Biol Chem. 1994 Jul 15;269(28):18259-62.
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Enzymatic transition states: thermodynamics, dynamics and analogue design.酶促过渡态：热力学、动力学与类似物设计
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