Sundberg R J, Rearick D E, Russell H F
J Pharm Sci. 1977 Feb;66(2):263-4. doi: 10.1002/jps.2600660231.
Several derivatives of 2-indolyl 5-(1,2,3,6-tetrahydropyridyl) ketone with various substituents on the pyridine nitrogen and with or without a benzenesulfonyl group on the indole nitrogen were synthesized and characterized by spectroscopic and analytical data. Only one showed erratic but confirmed activity in the P-388 screen. The other derivatives were inactive in the L-1210 leukemia screen.
合成了2-吲哚基5-(1,2,3,6-四氢吡啶基)酮的几种衍生物，这些衍生物在吡啶氮上带有各种取代基，吲哚氮上有或没有苯磺酰基，并通过光谱和分析数据进行了表征。只有一种在P-388筛选中显示出不稳定但已确认的活性。其他衍生物在L-1210白血病筛选中无活性。
