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Phosphodiesterase type IV inhibitors.

作者信息

Palfreyman M N, Souness J E

机构信息

Rhône-Poulence Rorer Central Research, Dagenham Research Centre, Essex, U.K.

出版信息

Prog Med Chem. 1996;33:1-52. doi: 10.1016/s0079-6468(08)70302-3.

DOI:10.1016/s0079-6468(08)70302-3
PMID:8776940
Abstract
摘要

相似文献

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Phosphodiesterase type IV inhibitors.磷酸二酯酶IV型抑制剂
Prog Med Chem. 1996;33:1-52. doi: 10.1016/s0079-6468(08)70302-3.
2
Isoenzyme selective phosphodiesterase inhibitors: potential clinical uses.同工酶选择性磷酸二酯酶抑制剂:潜在的临床用途。
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Isoenzyme-selective cyclic nucleotide phosphodiesterase inhibitors: effects on airways smooth muscle.同工酶选择性环核苷酸磷酸二酯酶抑制剂:对气道平滑肌的作用
Int J Biochem Cell Biol. 1995 Jan;27(1):29-37. doi: 10.1016/1357-2725(94)00060-3.
4
Immunomodulatory actions of xanthines and isoenzyme selective phosphodiesterase inhibitors.
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Effects of isozyme selective phosphodiesterase inhibitors on bovine tracheal smooth muscle tone.同工酶选择性磷酸二酯酶抑制剂对牛气管平滑肌张力的影响。
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6
Anti-inflammatory and bronchodilator properties of RP 73401, a novel and selective phosphodiesterase type IV inhibitor.新型选择性磷酸二酯酶IV型抑制剂RP 73401的抗炎及支气管扩张特性
Br J Pharmacol. 1994 Dec;113(4):1423-31. doi: 10.1111/j.1476-5381.1994.tb17156.x.
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Substituted pyrazolopyridines as potent and selective PDE5 inhibitors: potential agents for treatment of erectile dysfunction.
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Phosphodiesterase IV inhibitors synergistically potentiate relaxation induced by forskolin in guinea-pig trachea.
Clin Exp Pharmacol Physiol. 1998 Feb;25(2):114-9. doi: 10.1111/j.1440-1681.1998.tb02187.x.
9
The crystal structure, absolute configuration, and phosphodiesterase inhibitory activity of (+)-1-(4-bromobenzyl)-4-(3-(cyclopentyloxy)- 4-methoxyphenyl)-pyrrolidin-2-one.
J Med Chem. 1993 Oct 29;36(22):3274-7. doi: 10.1021/jm00074a007.
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Control of airway smooth muscle tone: II-pharmacology of relaxation.气道平滑肌张力的调控:II. 舒张药理学
Respir Med. 2000 Jun;94(6):519-28. doi: 10.1053/rmed.1999.0738.

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