Pharmacokinetics of isoniazid metabolism in man.

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作者信息

Ellard G A, Gammon P T

出版信息

J Pharmacokinet Biopharm. 1976 Apr;4(2):83-113. doi: 10.1007/BF01086149.

DOI:10.1007/BF01086149

PMID:950592

Abstract

摘要

相似文献

Pharmacokinetics of isoniazid metabolism in man.

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本文引用的文献

ASPECTS OF THE METABOLISM OF ISONIAZID AND ACETYLISONIAZID IN THE HUMAN AND THE DOG.

J Med Pharm Chem. 1962 Jan;5:196-203. doi: 10.1021/jm01236a019.

A study of the renal clearances, metabolic inactivation rates, and serum fall-off interaction of isoniazid and paraminosalicylic acid in man.人体中异烟肼和对氨基水杨酸的肾脏清除率、代谢失活率及血清衰减相互作用的研究。

Am Rev Respir Dis. 1961 Sep;84:371-8. doi: 10.1164/arrd.1961.84.3.371.

Further observations on the determination of the isoniazid inactivator phenotype.关于异烟肼灭活剂表型测定的进一步观察

Bull Johns Hopkins Hosp. 1961 Jan;108:60-6.

Acetylation of hydrazine and the formation of 1,2-diacetylhydrazine in vivo.

J Pharmacol Exp Ther. 1959 Jun;126(2):109-16.

Kinetic considerations relating to the accrual and elimination of drug metabolites.与药物代谢物的累积和消除相关的动力学考量。

Br J Pharmacol Chemother. 1967 Feb;29(2):136-49. doi: 10.1111/j.1476-5381.1967.tb01947.x.

Kinetics of competitive inhibition of salicylic acid conjugation with glycine in man.

Biochem Pharmacol. 1966 Aug;15(8):1033-8. doi: 10.1016/0006-2952(66)90267-x.

Comparative studies on the metabolism of isoniazid and isoniazid hydroazones in the dog.

Arch Int Pharmacodyn Ther. 1966 Feb;159(2):328-39.

Studies on the metabolic basis for the genetically determined capacities for isoniazid inactivation in man.

J Pharmacol Exp Ther. 1965 Nov;150(2):298-304.

Partial purification and properties of the isoniazid transacetylase in human liver. Its relationship to the acetylation of p-aminosalicylic acid.人肝脏中异烟肼转乙酰酶的部分纯化及性质。其与对氨基水杨酸乙酰化作用的关系。

J Clin Invest. 1965 Dec;44(12):1992-2002. doi: 10.1172/JCI105306.

The mechanism of isoniazid acetylation by human N-acetyltransferase.

Biochim Biophys Acta. 1968 Jan 8;151(1):276-8. doi: 10.1016/0005-2744(68)90184-8.

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