Han H, Yoon J, Janda K D
Department of Chemistry, Scripps Research Institute, La Jolla, CA, USA.
Bioorg Med Chem Lett. 1998 Jan 6;8(1):117-20. doi: 10.1016/s0960-894x(97)10198-6.
Solution syntheses of azapeptide pentamers 2, 3, and 4 were accomplished. The binding affinity of these azapeptides and azatide 1 were examined in the context of monoclonal antibody 3-E7 known to strongly bind the [Leu5]enkephalin sequence.