N-arylpiperazinone inhibitors of farnesyltransferase: discovery and biological activity.
作者信息
Williams T M, Bergman J M, Brashear K, Breslin M J, Dinsmore C J, Hutchinson J H, MacTough S C, Stump C A, Wei D D, Zartman C B, Bogusky M J, Culberson J C, Buser-Doepner C, Davide J, Greenberg I B, Hamilton K A, Koblan K S, Kohl N E, Liu D, Lobell R B, Mosser S D, O'Neill T J, Rands E, Schaber M D, Huff J R
机构信息
Department of Medicinal Chemistry, Merck Research Laboratories, West Point, Pennsylvania 19486, USA.
出版信息
J Med Chem. 1999 Sep 23;42(19):3779-84. doi: 10.1021/jm990254z.
PMID:10508426
Abstract
摘要
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