Zhang Xiaoxia, Campo Marino A, Yao Tuanli, Larock Richard C
Department of Chemistry, Iowa State University, Ames, IA 50011, USA.
Org Lett. 2005 Mar 3;7(5):763-6. doi: 10.1021/ol0476218.
Quinolines substituted in the 3-position by an iodo or phenylseleno group are readily prepared in good to excellent yields by the reaction of propargylic anilines with appropriate electrophiles under mild reaction conditions. [reaction: see text]
在温和的反应条件下，通过炔丙基苯胺与适当的亲电试剂反应，可轻松制备在3位被碘或苯硒基取代的喹啉，产率良好至优异。[反应：见正文]
