Derivatives of 2-mercaptobenzenesulphonamide. X. Synthesis of 1-dialkylaminoalkyl-2-(2-mercaptobenzenesulphonyl)guanidines with potential pharmacological activity.

Synthesis of 2-(4-R(1)-5-R(2)-2-mercaptobenzenesulphonyl)derivatives of 1-(dialkylaminoalkyl)-3-isobutylguanidine (III b-l) and 1,3-di(2-dialkylaminoethyl)guanidine (IV-V) as well as subsequent S-2-aminoethylation reaction VI a-h, VII a-b have been described.