Woodhouse Susan L, Ziolkowski Erin J, Rendina Louis M
School of Chemistry and Physics, The University of Adelaide, Adelaide, South Australia 5005, Australia.
Dalton Trans. 2005 Sep 7(17):2827-9. doi: 10.1039/b508340k. Epub 2005 Jul 25.
A series of novel, dinuclear (2,2':6',2''-terpyridine)platinum(ii) complexes containing bis(thioalkyl)-dicarba-closo-dodecaborane(12)(carborane) ligands were prepared and characterised, and their preliminary anti-cancer characteristics have been determined in vitro; the complexes are the first examples of bis-intercalator complexes containing a boron-rich carborane cage.
制备并表征了一系列含有双(硫代烷基)-二碳-闭式-十二硼烷(12)(碳硼烷)配体的新型双核(2,2':6',2''-三联吡啶)铂(II)配合物,并在体外测定了它们初步的抗癌特性;这些配合物是含有富硼碳硼烷笼的双嵌入剂配合物的首例。