1990年礼来奖讲座。一种看待激动作用和拮抗作用的方式：来自沙丁胺醇、沙美特罗及其他β-肾上腺素能受体激动剂的经验教训。 - Suppr

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超能文献

The 1990 Lilly Prize Lecture. A way of looking at agonism and antagonism: lessons from salbutamol, salmeterol and other beta-adrenoceptor agonists.

作者信息

Jack D

机构信息

Glaxo Holdings Limited, Ware, Hertfordshire.

出版信息

Br J Clin Pharmacol. 1991 May;31(5):501-14. doi: 10.1111/j.1365-2125.1991.tb05571.x.

DOI:10.1111/j.1365-2125.1991.tb05571.x

PMID:1679656

原文链接:https://pmc.ncbi.nlm.nih.gov/articles/PMC1368467/

Abstract

摘要

https://cdn.ncbi.nlm.nih.gov/pmc/blobs/254f/1368467/cc540b0513a8/brjclinpharm00058-0020-a.jpg

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本文引用的文献

A modification of receptor theory.受体理论的一种修正。

Br J Pharmacol Chemother. 1956 Dec;11(4):379-93. doi: 10.1111/j.1476-5381.1956.tb00006.x.

The technique of superfusion.超灌注技术。

Br J Pharmacol Chemother. 1953 Sep;8(3):321-6. doi: 10.1111/j.1476-5381.1953.tb00801.x.

Airway response to salbutamol: effect of regular salbutamol inhalations in normal, atopic, and asthmatic subjects.气道对沙丁胺醇的反应：正常、特应性和哮喘患者中规律吸入沙丁胺醇的效果。

Thorax. 1982 Apr;37(4):280-7. doi: 10.1136/thx.37.4.280.

Differentiation of receptors responsive to isoproterenol.对异丙肾上腺素产生反应的受体的分化

Life Sci. 1967 Nov 1;6(21):2241-9. doi: 10.1016/0024-3205(67)90031-8.

Differentiation of receptor systems activated by sympathomimetic amines.拟交感胺激活的受体系统的分化

Nature. 1967 May 6;214(5088):597-8. doi: 10.1038/214597a0.

Saligenin analogs of sympathomimetic catecholamines.拟交感神经儿茶酚胺的水杨苷类似物。

J Med Chem. 1970 Jul;13(4):674-80. doi: 10.1021/jm00298a022.

Adenyl cyclase as an adrenergic receptor.作为肾上腺素能受体的腺苷酸环化酶。

Ann N Y Acad Sci. 1967 Feb 10;139(3):703-23. doi: 10.1111/j.1749-6632.1967.tb41239.x.

The inducement of tone and its inhibition in isolated tracheal muscle.离体气管平滑肌中张力的诱导及其抑制

J Pharm Pharmacol. 1971 Mar;23(3):220-2. doi: 10.1111/j.2042-7158.1971.tb08648.x.

Recent beta-adrenoreceptor stimulants.近期的β-肾上腺素能受体兴奋剂。

Adv Drug Res. 1970;5:197-253.

Quinterenol, a new beta adrenergic stimulant.喹特罗醇，一种新型β肾上腺素能兴奋剂。

J Pharmacol Exp Ther. 1968 Jul;162(1):60-9.

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