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本文引用的文献

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Optimization of a series of potent and selective ketone histone deacetylase inhibitors.
Bioorg Med Chem Lett. 2008 Oct 15;18(20):5528-32. doi: 10.1016/j.bmcl.2008.09.003. Epub 2008 Sep 6.
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Enantioselective total synthesis of (+)-largazole, a potent inhibitor of histone deacetylase.
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Total synthesis and biological mode of action of largazole: a potent class I histone deacetylase inhibitor.
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A concise total synthesis of largazole, solution structure, and some preliminary structure activity relationships.
Org Lett. 2008 Aug 21;10(16):3595-8. doi: 10.1021/ol8013478. Epub 2008 Jul 11.
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Total synthesis and molecular target of largazole, a histone deacetylase inhibitor.
J Am Chem Soc. 2008 Jul 2;130(26):8455-9. doi: 10.1021/ja8013727. Epub 2008 May 29.
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Structural origin of selectivity in class II-selective histone deacetylase inhibitors.
J Med Chem. 2008 May 22;51(10):2898-906. doi: 10.1021/jm7015254. Epub 2008 Apr 16.
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Improved total synthesis of the potent HDAC inhibitor FK228 (FR-901228).
Org Lett. 2008 Feb 21;10(4):613-6. doi: 10.1021/ol702957z. Epub 2008 Jan 19.
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Structure and activity of largazole, a potent antiproliferative agent from the Floridian marine cyanobacterium Symploca sp.
J Am Chem Soc. 2008 Feb 13;130(6):1806-7. doi: 10.1021/ja7110064. Epub 2008 Jan 19.
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Fluorous-based small-molecule microarrays for the discovery of histone deacetylase inhibitors.
Angew Chem Int Ed Engl. 2007;46(42):7960-4. doi: 10.1002/anie.200703198.

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