生物膜中药物分子的结构分析 - Suppr

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Structural analysis of drug molecules in biological membranes.

作者信息

Herbette L G, Chester D W, Rhodes D G

出版信息

Biophys J. 1986 Jan;49(1):91-4. doi: 10.1016/S0006-3495(86)83605-0.

DOI:10.1016/S0006-3495(86)83605-0

PMID:19431663

原文链接:https://pmc.ncbi.nlm.nih.gov/articles/PMC1329589/

Abstract

摘要

https://cdn.ncbi.nlm.nih.gov/pmc/blobs/e125/1329589/4e72d7ad930c/biophysj00184-0101-a.jpg

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本文引用的文献

Crystal structures and pharmacological activity of calcium channel antagonists: 2,6-dimethyl-3,5-dicarbomethoxy-4-(unsubstituted, 2-methyl-, 4-methyl-, 3-nitro-, 4-nitro-, and 2,4-dinitrophenyl)-1,4-dihydropyridine.钙通道拮抗剂的晶体结构与药理活性：2,6 - 二甲基 - 3,5 - 二羧酸甲酯基 - 4 -（未取代、2 - 甲基、4 - 甲基、3 - 硝基、4 - 硝基以及2,4 - 二硝基苯基）- 1,4 - 二氢吡啶

J Med Chem. 1982 Feb;25(2):126-31. doi: 10.1021/jm00344a007.

Comparisons of the interaction of propranolol and timolol with model and biological membrane systems.普萘洛尔和噻吗洛尔与模型及生物膜系统相互作用的比较。

Mol Pharmacol. 1983 Sep;24(2):259-69.

Phospholipid asymmetry in the isolated sarcoplasmic reticulum membrane.分离的肌浆网膜中的磷脂不对称性。

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Sites of action of Ca2+ channel inhibitors.钙离子通道抑制剂的作用位点。

Biochem Pharmacol. 1983 Dec 1;32(23):3499-507. doi: 10.1016/0006-2952(83)90295-2.

Dihydropyridine derivatives prolong the open state of Ca channels in cultured cardiac cells.二氢吡啶衍生物可延长培养心肌细胞中钙通道的开放状态。

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