通过烯胺的分子内环化反应实现碘介导的 3H-吲哚合成。
Iodine-mediated synthesis of 3H-indoles via intramolecular cyclization of enamines.
机构信息
Department of Chemistry, Renmin University of China, Beijing 100872, China.
出版信息
J Org Chem. 2010 Jul 2;75(13):4636-9. doi: 10.1021/jo100796s.
PMID:20524670
Abstract
The synthesis of 3H-indoles was achieved via the iodine-mediated intramolecular cyclization of enamines. A wide variety of 3H-indole derivatives bearing multifunctional groups were obtained in good to high yields under transition metal-free reaction conditions.
摘要
通过碘介导的烯胺的分子内环化反应，实现了 3H-吲哚的合成。在无过渡金属反应条件下，以良好到高产率得到了多种带有多功能基团的 3H-吲哚衍生物。
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