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本文引用的文献

1
Irreversible inhibitors of c-Src kinase that target a nonconserved cysteine.
ACS Chem Biol. 2012 Nov 16;7(11):1910-7. doi: 10.1021/cb300337u. Epub 2012 Sep 5.
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Highly specific, bisubstrate-competitive Src inhibitors from DNA-templated macrocycles.
Nat Chem Biol. 2012 Feb 19;8(4):366-74. doi: 10.1038/nchembio.792.
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How chemoproteomics can enable drug discovery and development.
Chem Biol. 2012 Jan 27;19(1):11-22. doi: 10.1016/j.chembiol.2012.01.001.
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In situ kinase profiling reveals functionally relevant properties of native kinases.
Chem Biol. 2011 Jun 24;18(6):699-710. doi: 10.1016/j.chembiol.2011.04.011.
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The resurgence of covalent drugs.
Nat Rev Drug Discov. 2011 Apr;10(4):307-17. doi: 10.1038/nrd3410.
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A structure-guided approach to creating covalent FGFR inhibitors.
Chem Biol. 2010 Mar 26;17(3):285-95. doi: 10.1016/j.chembiol.2010.02.007.
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Src kinases as therapeutic targets for cancer.
Nat Rev Clin Oncol. 2009 Oct;6(10):587-95. doi: 10.1038/nrclinonc.2009.129.
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Global target profile of the kinase inhibitor bosutinib in primary chronic myeloid leukemia cells.
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Small molecule inhibitors of Lck: the search for specificity within a kinase family.
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