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N,N-disubstituted 2-aminothiazolines as new inhibitors of serine esterases.

作者信息

Boltneva N P, Serebryakova O G, Makhaeva G F, Serkov I V, Proshin A N, Bachurin S O

机构信息

Institute of Physiologically Active Substances, Russian Academy of Sciences, Chernogolovka, Moscow oblast, 142432, Russia.

出版信息

Dokl Biochem Biophys. 2013 Jul-Aug;451:209-11. doi: 10.1134/S160767291304011X. Epub 2013 Aug 23.

DOI:10.1134/S160767291304011X
PMID:23975403
Abstract
摘要

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本文引用的文献

1
Organophosphorus compound esterase profiles as predictors of therapeutic and toxic effects.有机磷化合物酯酶谱作为治疗和毒性效应的预测指标。
Chem Biol Interact. 2013 Mar 25;203(1):231-7. doi: 10.1016/j.cbi.2012.10.012. Epub 2012 Nov 2.
2
Esterase profile of O-phosphorylated ethyltrifluorolactates in prediction of their therapeutic and toxic effects.
Dokl Biochem Biophys. 2012 Mar-Apr;443:81-5. doi: 10.1134/S1607672912020068. Epub 2012 May 5.
3
Esterase profile and analysis of structure-inhibitor selectivity relationships for homologous phosphorylated 1-hydroperfluoroisopropanols.同源磷酸化1-氢全氟异丙醇的酯酶谱及结构-抑制剂选择性关系分析
Dokl Biochem Biophys. 2008 Nov-Dec;423:352-7. doi: 10.1134/s1607672908060094.
4
Overview of the chemistry of 2-thiazolines.2-噻唑啉的化学概述。
Chem Rev. 2009 Mar 11;109(3):1371-401. doi: 10.1021/cr800189z.
5
Recent developments in cholinesterases inhibitors for Alzheimer's disease treatment.用于治疗阿尔茨海默病的胆碱酯酶抑制剂的最新进展。
Curr Med Chem. 2007;14(25):2654-79. doi: 10.2174/092986707782023217.
6
Chemiluminescent high-throughput microassay applied to imidazo[2,1-b]thiazole derivatives as potential acetylcholinesterase and butyrylcholinesterase inhibitors.化学发光高通量微量分析用于咪唑并[2,1-b]噻唑衍生物作为潜在的乙酰胆碱酯酶和丁酰胆碱酯酶抑制剂的研究
Eur J Med Chem. 2008 Mar;43(3):657-61. doi: 10.1016/j.ejmech.2007.04.018. Epub 2007 May 21.
7
Novel structural motifs consisting of chiral thiazolines: synthesis, molecular recognition, and anticancer activity.由手性噻唑啉组成的新型结构基序：合成、分子识别及抗癌活性
Chemistry. 2007;13(11):3026-38. doi: 10.1002/chem.200601446.
8
Carboxylesterases--detoxifying enzymes and targets for drug therapy.羧酸酯酶——解毒酶及药物治疗靶点
Curr Med Chem. 2006;13(9):1045-54. doi: 10.2174/092986706776360969.
9
Cholinesterase inhibitors: new roles and therapeutic alternatives.胆碱酯酶抑制剂：新作用及治疗选择
Pharmacol Res. 2004 Oct;50(4):433-40. doi: 10.1016/j.phrs.2003.11.017.
10
Competitive inhibition of acetylcholinesterase by several thiazolines and oxazolines.
Arch Biochem Biophys. 1960 Aug;89:293-5. doi: 10.1016/0003-9861(60)90057-6.