Li Jian, Wang Hongni, Sun Jiangtao, Yang Yang, Liu Li
School of Pharmaceutical Engineering & Life Sciences, Chang Zhou University, Changzhou, 213164, P. R. China.
Org Biomol Chem. 2014 Apr 28;12(16):2523-7. doi: 10.1039/c3ob42431f.
A mild gold-catalyzed three-component dehydrogenative coupling of terminal alkynes to amines and indole-2-carboxaldehyde has been developed, which provides a practical synthetic strategy for the synthesis of indole derivatives.
已开发出一种温和的金催化末端炔烃与胺和吲哚 -2-甲醛的三组分脱氢偶联反应,该反应为吲哚衍生物的合成提供了一种实用的合成策略。