College of Chemistry and Pharmaceutical Sciences, Qingdao Agricultural University , Qingdao 266109, China.
Org Lett. 2017 Nov 3;19(21):5724-5727. doi: 10.1021/acs.orglett.7b02294.
The organocatalytic alkylation of 2-methyl-N-heteroaromatics with alcohols has been achieved via S1-type C(sp)-H functionalization, providing a green and efficient synthesis of indole and ferrocene-functionalized N-heteroaromatics in high yields.
通过 S1 型 C(sp3)-H 官能化反应，实现了 2-甲基-N-杂芳烃与醇的有机催化烷基化反应，为吲哚和二茂铁基 N-杂芳烃的高效绿色合成提供了一种新方法，产率很高。
