College of Chemistry and Chemical Engineering, Nantong University, Nantong 226019, China.
School of Environmental and Chemical Engineering, Jiangsu University of Science and Technology, Zhenjiang 212003, China.
Molecules. 2017 Nov 27;22(12):2000. doi: 10.3390/molecules22122000.
In this study, in order to find novel biologically active pyrazole oxime derivatives, twenty-eight new pyrazole oxime compounds containing a substituted isoxazole ring were synthesized and evaluated for their acaricidaland insecticidal activities. Bioassays exhibited that some target compounds indicated good acaricidal and insecticidal activities against , , , and . Especially, compounds , , , and showed 100.00%, 90.56%, 90.78%, and 90.62% insecticidal activities against at the concentration of 20 μg/mL, respectively, compounds and had 70.86% and 100.00% insecticidal activities against at 20 μg/mL, respectively.
在这项研究中，为了寻找新型具有生物活性的吡唑肟衍生物，合成了 28 种新型含取代异恶唑环的吡唑肟化合物，并对其杀螨和杀虫活性进行了评价。生物测定结果表明，部分目标化合物对 、 、 、 表现出良好的杀螨和杀虫活性。特别是化合物 、 、 、 对 浓度为 20μg/mL 时的杀虫活性分别为 100.00%、90.56%、90.78%和 90.62%，化合物 和 对 20μg/mL 时的杀虫活性分别为 70.86%和 100.00%。
