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四氢喹啉化学进展。

Progress in the Chemistry of Tetrahydroquinolines.

机构信息

Department of Chemistry, School of Chemical and Biotechnology , SASTRA Deemed University , Thanjavur 613401 , Tamil Nadu , India.

Department of Chemistry and Chemical Sciences , Central University of Jammu , Rahya-Suchani (Bagla) , District-Samba, Jammu 181143 , Jammu and Kashmir , India.

出版信息

Chem Rev. 2019 Apr 24;119(8):5057-5191. doi: 10.1021/acs.chemrev.8b00567. Epub 2019 Apr 9.

DOI:10.1021/acs.chemrev.8b00567
PMID:30963764
Abstract

Tetrahydroquinoline is one of the most important simple nitrogen heterocycles, being widespread in nature and present in a broad variety of pharmacologically active compounds. This Review summarizes the progress achieved in the chemistry of tetrahydroquinolines, with emphasis on their synthesis, during the period from mid-2010 to early 2018.

摘要

四氢喹啉是最重要的简单氮杂环之一,在自然界中广泛存在,并存在于多种具有药理活性的化合物中。本文综述了 2010 年年中至 2018 年初期间四氢喹啉化学的进展,重点介绍了它们的合成。

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