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Evaluation of Potential Therapeutic Options for COVID-19.

作者信息

Austin Daren, Okour Malek

机构信息

Clinical Pharmacology Modelling & Simulation, GlaxoSmithKline Research & Development, Collegeville, Pennsylvania, USA.

出版信息

J Clin Pharmacol. 2020 Aug;60(8):976-977. doi: 10.1002/jcph.1669. Epub 2020 Jul 8.

DOI:10.1002/jcph.1669
PMID:32469418
原文链接:https://pmc.ncbi.nlm.nih.gov/articles/PMC7283735/
Abstract
摘要

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Identification of Antiviral Drug Candidates against SARS-CoV-2 from FDA-Approved Drugs.从 FDA 批准药物中鉴定抗 SARS-CoV-2 的抗病毒候选药物。
Antimicrob Agents Chemother. 2020 Jun 23;64(7). doi: 10.1128/AAC.00819-20.
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The FDA-approved drug ivermectin inhibits the replication of SARS-CoV-2 in vitro.美国食品药品监督管理局批准的药物伊维菌素可抑制 SARS-CoV-2 的体外复制。
Antiviral Res. 2020 Jun;178:104787. doi: 10.1016/j.antiviral.2020.104787. Epub 2020 Apr 3.
3
In Vitro Antiviral Activity and Projection of Optimized Dosing Design of Hydroxychloroquine for the Treatment of Severe Acute Respiratory Syndrome Coronavirus 2 (SARS-CoV-2).羟氯喹治疗严重急性呼吸综合征冠状病毒 2 (SARS-CoV-2)的体外抗病毒活性和优化剂量设计预测。
Clin Infect Dis. 2020 Jul 28;71(15):732-739. doi: 10.1093/cid/ciaa237.
4
Remdesivir and chloroquine effectively inhibit the recently emerged novel coronavirus (2019-nCoV) in vitro.瑞德西韦和氯喹在体外能有效抑制新出现的新型冠状病毒(2019 - 新冠病毒)。
Cell Res. 2020 Mar;30(3):269-271. doi: 10.1038/s41422-020-0282-0. Epub 2020 Feb 4.
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Pharmacokinetics/pharmacodynamics of chloroquine and artemisinin-based combination therapy with primaquine.氯喹和青蒿素类联合治疗与伯氨喹的药代动力学/药效学。
Malar J. 2019 Sep 23;18(1):325. doi: 10.1186/s12936-019-2950-4.
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A phase I study of niclosamide in combination with enzalutamide in men with castration-resistant prostate cancer.尼氯硝唑联合恩扎卢胺治疗去势抵抗性前列腺癌的 I 期研究。
PLoS One. 2018 Jun 1;13(6):e0198389. doi: 10.1371/journal.pone.0198389. eCollection 2018.
7
Favipiravir pharmacokinetics in Ebola-Infected patients of the JIKI trial reveals concentrations lower than targeted.JIKI试验中埃博拉感染患者的法匹拉韦药代动力学显示浓度低于目标值。
PLoS Negl Trop Dis. 2017 Feb 23;11(2):e0005389. doi: 10.1371/journal.pntd.0005389. eCollection 2017 Feb.
8
Pharmacokinetics of hydroxychloroquine and its clinical implications in chemoprophylaxis against malaria caused by Plasmodium vivax.羟氯喹的药代动力学及其在间日疟原虫所致疟疾化学预防中的临床意义
Antimicrob Agents Chemother. 2009 Apr;53(4):1468-75. doi: 10.1128/AAC.00339-08. Epub 2009 Feb 2.
9
Safety, tolerability, and pharmacokinetics of escalating high doses of ivermectin in healthy adult subjects.健康成年受试者中递增高剂量伊维菌素的安全性、耐受性和药代动力学。
J Clin Pharmacol. 2002 Oct;42(10):1122-33. doi: 10.1177/009127002401382731.
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The tolerance to and pharmacokinetics of penciclovir (BRL 39,123A), a novel antiherpes agent, administered by intravenous infusion to healthy subjects.新型抗疱疹药物喷昔洛韦(BRL 39,123A)静脉输注健康受试者后的耐受性及药代动力学。
Eur J Clin Pharmacol. 1992;43(5):513-6. doi: 10.1007/BF02285093.