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无溶剂法合成炔丙胺：综述

Solvent-free synthesis of propargylamines: an overview.

作者信息

Manujyothi Ravi, Aneeja Thaipparambil, Anilkumar Gopinathan

机构信息

Institute for Integrated Programmes and Research in Basic Sciences (IIRBS), Mahatma Gandhi University Priyadarsini Hills P O Kottayam Kerala 686560 India

School of Chemical Sciences, Mahatma Gandhi University Priyadarsini Hills P O Kottayam Kerala 686560 India.

出版信息

RSC Adv. 2021 May 30;11(32):19433-19449. doi: 10.1039/d1ra03324g. eCollection 2021 May 27.

DOI:10.1039/d1ra03324g
PMID:35479216
原文链接:https://pmc.ncbi.nlm.nih.gov/articles/PMC9033675/
Abstract

Propargylamines are a class of compounds with many pharmaceutical and biological properties. A green approach to synthesize such compounds is very relevant. This review aims to describe the solvent-free synthetic approaches towards propargylamines A and KA coupling reactions covering the literature up to 2021.

摘要

炔丙胺是一类具有多种药物和生物学特性的化合物。一种绿色的合成此类化合物的方法非常重要。本综述旨在描述截至2021年文献中关于炔丙胺A和KA偶联反应的无溶剂合成方法。

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