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The biological activity and the binding affinity of modified insulins determined on isolated rat fat cells.

作者信息

Gliemann J, Gammeltoft S

出版信息

Diabetologia. 1974 Apr;10(2):105-13. doi: 10.1007/BF01219665.

DOI:10.1007/BF01219665
PMID:4367434
Abstract
摘要

相似文献

1
The biological activity and the binding affinity of modified insulins determined on isolated rat fat cells.在分离的大鼠脂肪细胞上测定修饰胰岛素的生物活性和结合亲和力。
Diabetologia. 1974 Apr;10(2):105-13. doi: 10.1007/BF01219665.
2
Lipogenesis and insulin sensitivity of single fat cells.单个脂肪细胞的脂肪生成与胰岛素敏感性
J Physiol. 1974 Feb;236(3):499-516. doi: 10.1113/jphysiol.1974.sp010449.
3
Time course of insulin-receptor binding and insulin-induced lipogenesis in isolated rat fat cells.分离的大鼠脂肪细胞中胰岛素受体结合及胰岛素诱导的脂肪生成的时间进程。
J Biol Chem. 1975 May 10;250(9):3368-74.
4
Adenosine triphosphate-dependent inhibition of insulin-stimulated glucose transport in fat cells. Possible role of membrane phosphorylation.三磷酸腺苷依赖性抑制脂肪细胞中胰岛素刺激的葡萄糖转运。膜磷酸化的可能作用。
J Biol Chem. 1974 May 25;249(10):3170-80.
5
Insulin receptors in fat cells: relationship between binding and activation.脂肪细胞中的胰岛素受体:结合与激活之间的关系
Isr J Med Sci. 1975 Jul;11(7):656-63.
6
Insulin and microtubules in rat adipocytes.大鼠脂肪细胞中的胰岛素与微管
Science. 1971 Apr 16;172(3980):269-71. doi: 10.1126/science.172.3980.269.
7
Common mechanism of action of somatomedin and insulin on fat cells. Further evidence.生长调节素与胰岛素对脂肪细胞的共同作用机制。进一步的证据。
Isr J Med Sci. 1974 Oct;10(10):1254-62.
8
The insulin-like activity of cyclic nucleotides and their inhibition by caffeine on the isolated fat cells.环核苷酸的胰岛素样活性及其在分离脂肪细胞中被咖啡因的抑制作用。
Biochem Biophys Res Commun. 1970;39(6):1065-72. doi: 10.1016/0006-291x(70)90667-4.
9
Nonsuppressible insulin-like activity: biological activity and receptor binding.非抑制性胰岛素样活性:生物活性与受体结合
Isr J Med Sci. 1975 Jul;11(7):664-78.
10
A simple free fat cell bioassay for insulin.一种用于胰岛素的简单游离脂肪细胞生物测定法。
Horm Metab Res. 1974 Jan;6(1):12-6. doi: 10.1055/s-0028-1093895.

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Fully dissolved glucose-responsive insulin delivery system based on a self-immolative insulin prodrug and glucose oxidase.基于自牺牲胰岛素前药和葡萄糖氧化酶的完全溶解的葡萄糖响应性胰岛素递送系统。
Chem Sci. 2025 Aug 11. doi: 10.1039/d5sc02817e.
2
An Investigation into the Acidity-Induced Insulin Agglomeration: Implications for Drug Delivery and Translation.酸度诱导胰岛素聚集的研究:对药物递送及转化的启示
ACS Omega. 2023 Jul 6;8(28):25279-25287. doi: 10.1021/acsomega.3c02482. eCollection 2023 Jul 18.
3
Amyloid Fibrillation of Insulin: Amelioration Strategies and Implications for Translation.

本文引用的文献

1
Action of carboxypeptidase- A on bovine insulin: preparation of desalanine-desasparagine-insulin.羧肽酶A对牛胰岛素的作用:去丙氨酸-去天冬酰胺胰岛素的制备
Biochemistry. 1963 Jan-Feb;2:16-22. doi: 10.1021/bi00901a004.
2
Intramolecular cross-linked insulin.分子内交联胰岛素
FEBS Lett. 1972 Mar;21(1):105-108. doi: 10.1016/0014-5793(72)80175-3.
3
Kinetics of 125I-insulin binding to rat liver plasma membranes.125I标记胰岛素与大鼠肝细胞膜结合的动力学
胰岛素的淀粉样纤维化:改善策略及其转化意义
ACS Pharmacol Transl Sci. 2022 Oct 12;5(11):1050-1061. doi: 10.1021/acsptsci.2c00174. eCollection 2022 Nov 11.
4
Smart Thermosensitive Copolymer Incorporating Chitosan-Zinc-Insulin Electrostatic Complexes for Controlled Delivery of Insulin: Effect of Chitosan Chain Length.用于胰岛素控释的含壳聚糖-锌-胰岛素静电复合物的智能热敏共聚物:壳聚糖链长的影响
Int J Polym Mater. 2020;69(16):1054-1068. doi: 10.1080/00914037.2019.1655750. Epub 2019 Aug 26.
5
Site-Specific Insulin-Trehalose Glycopolymer Conjugate by Grafting From Strategy Improves Bioactivity.通过接枝策略制备的位点特异性胰岛素-海藻糖糖聚合物缀合物可提高生物活性。
ACS Macro Lett. 2018 Mar 20;7(3):324-329. doi: 10.1021/acsmacrolett.7b00974. Epub 2018 Feb 20.
6
Oxidation of therapeutic proteins and peptides: structural and biological consequences.治疗性蛋白质和肽的氧化:结构和生物学后果
Pharm Res. 2014 Mar;31(3):541-53. doi: 10.1007/s11095-013-1199-9. Epub 2013 Sep 25.
7
Design of an active ultrastable single-chain insulin analog: synthesis, structure, and therapeutic implications.活性超稳定单链胰岛素类似物的设计:合成、结构及治疗意义
J Biol Chem. 2008 May 23;283(21):14703-16. doi: 10.1074/jbc.M800313200. Epub 2008 Mar 10.
8
Human insulin production from a novel mini-proinsulin which has high receptor-binding activity.源自具有高受体结合活性的新型微型胰岛素原的人胰岛素生产。
Biochem J. 1998 Feb 1;329 ( Pt 3)(Pt 3):631-5. doi: 10.1042/bj3290631.
9
Inactive conformation of an insulin despite its wild-type sequence.尽管胰岛素具有野生型序列,但处于无活性构象。
Protein Sci. 1997 Mar;6(3):580-7. doi: 10.1002/pro.5560060307.
10
Solution structure of a mini IGF-1.一种小型胰岛素样生长因子-1(IGF-1)的溶液结构
Protein Sci. 1996 Nov;5(11):2193-202. doi: 10.1002/pro.5560051106.
FEBS Lett. 1971 Sep 1;16(4):339-342. doi: 10.1016/0014-5793(71)80385-x.
4
Preparation and characterization of desoctapeptide-insulin.去八肽胰岛素的制备与表征
Biochim Biophys Acta. 1967 Feb 21;133(2):219-23. doi: 10.1016/0005-2795(67)90061-x.
5
Immunology conformation and biological activity of insulin.胰岛素的免疫学构象与生物学活性。
Diabetes. 1969 Apr;18(4):193-205. doi: 10.2337/diab.18.4.193.
6
[Des-PheB1-insulin, a crystalline analogue of bovine insulin].[去苯丙氨酸B1胰岛素,一种牛胰岛素的晶体类似物]
Hoppe Seylers Z Physiol Chem. 1969 Jun;350(6):741-50. doi: 10.1515/bchm2.1969.350.1.741.
7
The effect of chemical modifications induced in insulin on the reactivity of the interchain disulphide bonds towards sodium sulphite.胰岛素中诱导的化学修饰对链间二硫键与亚硫酸钠反应活性的影响。
Biochem J. 1968 Jun;108(2):247-55. doi: 10.1042/bj1080247.
8
[Structure and action of insulin. 3. Synthetic A-chains with varied sequence].[胰岛素的结构与作用。3. 具有不同序列的合成A链]
Hoppe Seylers Z Physiol Chem. 1968 Apr;349(4):512-4.
9
[Structure and action of insulin. II. Synthetic A-chains with varied sequence].[胰岛素的结构与作用。II. 具有不同序列的合成A链]
Hoppe Seylers Z Physiol Chem. 1967 Dec;348(12):1715-7.
10
Assay of insulin-like activity by the isolated fat cell method. I. Factors influencing the response to crystalline insulin.用分离脂肪细胞法测定胰岛素样活性。I. 影响对结晶胰岛素反应的因素。
Diabetologia. 1967 Aug;3(4):382-8. doi: 10.1007/BF02342631.