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Sudoxicam and related N-heterocyclic carboxamides of 4-hydroxy-2H-1,2-benzothiazine 1,1-dioxide. Potent nonsteroidal antiinflammatory agents.

作者信息

Lombardino J G, Wiseman E H

出版信息

J Med Chem. 1972 Aug;15(8):848-9. doi: 10.1021/jm00278a016.

DOI:10.1021/jm00278a016
PMID:4625532
Abstract
摘要

相似文献

1
Sudoxicam and related N-heterocyclic carboxamides of 4-hydroxy-2H-1,2-benzothiazine 1,1-dioxide. Potent nonsteroidal antiinflammatory agents.舒多昔康及相关的4-羟基-2H-1,2-苯并噻嗪1,1-二氧化物的N-杂环羧酰胺。强效非甾体抗炎药。
J Med Chem. 1972 Aug;15(8):848-9. doi: 10.1021/jm00278a016.
2
Potent anti-inflammatory N-heterocyclic 3-carboxamides of 4-hydroxy-2-methyl-2H-1,2-benzothiazine 1,1-dioxide.
J Med Chem. 1973 May;16(5):493-6. doi: 10.1021/jm00263a017.
3
Anti-inflammatory and pharmacokinetic properties of sudoxicam N-(2-thiazolyl)-4-hydroxy-2-methyl-2H-1,2-benzothiazine-3-carboxamide 1,1-dioxide.
Biochem Pharmacol. 1972 Sep 1;21(17):2323-34. doi: 10.1016/0006-2952(72)90383-8.
4
Synthesis and antiinflammatory activity of some 3-carboxamides of 2-alkyl-4-hydroxy-2H-1,2-benzothiazine 1,1-dioxide.
J Med Chem. 1971 Dec;14(12):1171-5. doi: 10.1021/jm00294a008.
5
Excretion and metabolism of a nonsteroidal antiinflammatory agent, 4-hydroxy-2-methyl-2H-1,2-benzothiazine-3-carboxanilide 1,1-dioxide, in rat, dog, monkey, and man.
J Med Chem. 1971 Dec;14(12):1175-7. doi: 10.1021/jm00294a009.
6
1,2-benzothiazines. 6. 3-Carbamoyl-4-hydroxy-2H-1,2-benzothiazine 1,1-dioxides as antiinflammatory agents.
J Med Chem. 1973 Jan;16(1):44-8. doi: 10.1021/jm00259a013.
7
Synthesis and antiinflammatory evaluation of certain 5-akloxy-2,7-dialkyltryptamines.某些5-烷氧基-2,7-二烷基色胺的合成与抗炎活性评价
J Med Chem. 1973 Jul;16(7):757-65. doi: 10.1021/jm00265a004.
8
2-Phenyl-4H-cyclopentathiazole-4-carboxylic acids as potential antiinflammatory agents.2-苯基-4H-环戊并噻唑-4-羧酸作为潜在的抗炎剂。
J Med Chem. 1972 Aug;15(8):850-1. doi: 10.1021/jm00278a018.
9
Derivatives of indole-1-acetic acid as antiinflammatory agents.吲哚 - 1 - 乙酸衍生物作为抗炎剂。
J Med Chem. 1972 Oct;15(10):1081-2. doi: 10.1021/jm00280a027.
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Antiinflammatory 3,4-dihydro-2-alkyl-3-oxo-2H-1,2-benzothiazine-4-carboxamide 1,1-dioxides.
J Med Chem. 1971 Oct;14(10):973-7. doi: 10.1021/jm00292a022.

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