Synthesis and antiinflammatory activity of some 3-carboxamides of 2-alkyl-4-hydroxy-2H-1,2-benzothiazine 1,1-dioxide.

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作者信息

Lombardino J G, Wiseman E H, McLamore W M

出版信息

J Med Chem. 1971 Dec;14(12):1171-5. doi: 10.1021/jm00294a008.

DOI:10.1021/jm00294a008

PMID:5116229

Abstract

摘要

相似文献

Synthesis and antiinflammatory activity of some 3-carboxamides of 2-alkyl-4-hydroxy-2H-1,2-benzothiazine 1,1-dioxide.

J Med Chem. 1971 Dec;14(12):1171-5. doi: 10.1021/jm00294a008.

Potent anti-inflammatory N-heterocyclic 3-carboxamides of 4-hydroxy-2-methyl-2H-1,2-benzothiazine 1,1-dioxide.

J Med Chem. 1973 May;16(5):493-6. doi: 10.1021/jm00263a017.

Sudoxicam and related N-heterocyclic carboxamides of 4-hydroxy-2H-1,2-benzothiazine 1,1-dioxide. Potent nonsteroidal antiinflammatory agents.舒多昔康及相关的4-羟基-2H-1,2-苯并噻嗪1,1-二氧化物的N-杂环羧酰胺。强效非甾体抗炎药。

J Med Chem. 1972 Aug;15(8):848-9. doi: 10.1021/jm00278a016.

Antiinflammatory 3,4-dihydro-2-alkyl-3-oxo-2H-1,2-benzothiazine-4-carboxamide 1,1-dioxides.

J Med Chem. 1971 Oct;14(10):973-7. doi: 10.1021/jm00292a022.

1,2-benzothiazines. 6. 3-Carbamoyl-4-hydroxy-2H-1,2-benzothiazine 1,1-dioxides as antiinflammatory agents.

J Med Chem. 1973 Jan;16(1):44-8. doi: 10.1021/jm00259a013.

4-(3-(Dimethylamino)propyl)-3,4-dihydro-2-(1-hydroxyethyl)-3-phenyl-2H-1,4-benzothiazine and related compounds. A new class of antiinflammatory agents.

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[Synthesis and antiinflammatory activity of various 1,4-benzothiazine derivatives].

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[Synthesis and pharmacologic activity of the carboxamides of pyrazolo-1,2-benzothiazine and isoxazolo-1,2-benzothiazine (I)].吡唑并[1,2 - b]苯并噻嗪和异恶唑并[1,2 - b]苯并噻嗪羧酰胺的合成及药理活性（I）

Farmaco Sci. 1983 Jan;38(1):35-44.

Anti-inflammatory and pharmacokinetic properties of sudoxicam N-(2-thiazolyl)-4-hydroxy-2-methyl-2H-1,2-benzothiazine-3-carboxamide 1,1-dioxide.

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