Structure-activity studies leading to ethambutol, a new type of antituberculous compound.

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作者信息

Shepherd R G, Baughn C, Cantrall M L, Goodstein B, Thomas J P, Wilkinson R G

出版信息

Ann N Y Acad Sci. 1966 Apr 20;135(2):686-710. doi: 10.1111/j.1749-6632.1966.tb45516.x.

DOI:10.1111/j.1749-6632.1966.tb45516.x

PMID:5220237

Abstract

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相似文献

Structure-activity studies leading to ethambutol, a new type of antituberculous compound.

Ann N Y Acad Sci. 1966 Apr 20;135(2):686-710. doi: 10.1111/j.1749-6632.1966.tb45516.x.

[Cyclic analogs of ethambutol with antimycobacterial activity].

Farmaco Sci. 1983 Feb;38(2):73-80.

A new synthetic compound with antituberculous activity in mice: ethambutol (dextro-2,2'-(ethylenediimino)-di-l-butanol).一种在小鼠中具有抗结核活性的新型合成化合物：乙胺丁醇（右旋-2,2'-（乙二胺基）-二-1-丁醇）。

Am Rev Respir Dis. 1961 Jun;83:891-3. doi: 10.1164/arrd.1961.83.6.891.

[Microcrystallographic identification of a tuberculostatic: ethambutol, 2HCl].[一种抗结核药的微晶鉴定：盐酸乙胺丁醇]

J Pharm Belg. 1984 Jul-Aug;39(4):243-5.

[Some aspects of determination of the sensitivity of Mycobacterium tuberculosis to ethambutol using a semiliquid medium].[使用半液体培养基测定结核分枝杆菌对乙胺丁醇敏感性的某些方面]

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Characterization of the embB gene in Mycobacterium tuberculosis isolates from Barcelona and rapid detection of main mutations related to ethambutol resistance using a low-density DNA array-authors' response.巴塞罗那结核分枝杆菌分离株中embB基因的特征分析及使用低密度DNA芯片快速检测与乙胺丁醇耐药相关的主要突变——作者回应

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Growth inhibition of tubercle bacilli after pulsed exposures to combinations of antituberculous drugs.

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[Bacteriostatic effect of ethambutol on tubercle bacilli sensitive or resistant to other antitubercular drugs. A modification of the vertical diffusion method for determination of biologically active ethambutol].

Gruzlica. 1969 Jul;37(7):623-8.

Synthesis and biological evaluation of conformationally constrained analogues of the antitubercular agent ethambutol.抗结核药物乙胺丁醇构象受限类似物的合成与生物学评价

Bioorg Med Chem. 2007 Sep 1;15(17):5866-76. doi: 10.1016/j.bmc.2007.05.064. Epub 2007 Jun 2.

[ANTITUBERCULOUS ACTIVITY OF DEXTRO-2,2'-(ETHYLENEDIIMINO)-DI-1-BUTANOL (ETHAMBUTOL). (II) COMBINED EFFECT OF ETHAMBUTOL AND ISONIAZID].右旋-2,2'-（乙二胺基）-二-1-丁醇（乙胺丁醇）的抗结核活性。（II）乙胺丁醇与异烟肼的联合效应

Kekkaku. 1964 Jun;39:191-6.

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