氨基取代对4-溴苯乙醇胺β-肾上腺素能受体活性的影响。
The effect of amino-substitution on the beta-adrenoceptor activity of 4-bromophenylethanolamines.
作者信息
Letts L G, Temple D M, Orr A J, Williams L R
出版信息
Arch Int Pharmacodyn Ther. 1980 May;245(1):48-55.
PMID:6250504
Abstract
A series of 4-bromophenylethanolamines with a variety of amino substituents has been prepared. A detailed pharmacological evaluation has been made of their beta-adrenergic activity to study how the amino substituent may effect the mixed agonist and antagonist action of a phenylethanolamine series.
摘要
已制备了一系列带有各种氨基取代基的4-溴苯乙醇胺。对它们的β-肾上腺素能活性进行了详细的药理学评估，以研究氨基取代基如何影响苯乙醇胺系列的混合激动剂和拮抗剂作用。
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