Synthesis and pharmacological activity of 3-substituted pyrido[3',2':4,5]thieno[3,2-d]pyrimidin-4(3H)-ones.
作者信息
Bousquet E, Guerrera F, Siracusa M A, Caruso A, Amico-Roxas M
出版信息
Farmaco Sci. 1984 Feb;39(2):110-9. doi: 10.1002/chin.198435236.
PMID:6609089
Abstract
A series of 3-substituted pyridothienopyrimidin-4(3H)-ones has been synthesized from 2,7,9-trimethyl-4H-pyrido[3',2':4,5]thieno-[3,2-d] [ 1,3]oxazin-4-one. These compounds have been evaluated for analgesic, anti-inflammatory and antipyretic activities. The ulcerogenic effect of the compounds has been also studied.
摘要
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