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Novel method of estimating volume of distribution of a drug obeying Michaelis-Menten elimination kinetics.

作者信息

Lin Y J, Weidler D J, Garg D C, Wagner J G

出版信息

J Pharmacokinet Biopharm. 1978 Jun;6(3):197-207. doi: 10.1007/BF01312262.

DOI:10.1007/BF01312262
PMID:671226
Abstract
摘要

相似文献

1
Novel method of estimating volume of distribution of a drug obeying Michaelis-Menten elimination kinetics.
J Pharmacokinet Biopharm. 1978 Jun;6(3):197-207. doi: 10.1007/BF01312262.
2
New and simple method to predict dosage of drugs obeying simple Michaelis-Menten elimination kinetics and to distinguish such kinetics from simple first order and from parallel Michaelis-Menten and first order kinetics.预测遵循简单米氏消除动力学的药物剂量并将这种动力学与简单一级动力学、平行米氏动力学和一级动力学相区分的新的简单方法。
Ther Drug Monit. 1985;7(4):377-86. doi: 10.1097/00007691-198512000-00003.
3
Time to reach steady state and prediction of steady-state concentrations for drugs obeying Michaelis-Menten elimination kinetics.
J Pharmacokinet Biopharm. 1978 Jun;6(3):209-25. doi: 10.1007/BF01312263.
4
First-pass effect: nonlinear concept comprising an explicit solution of integrated Michaelis-Menten equation.首过效应:非线性概念,包含米氏方程积分的显式解。
J Pharm Sci. 1981 Feb;70(2):195-8. doi: 10.1002/jps.2600700221.
5
[Mathematical study on characteristics of the average steady-state for drugs obeying Michaelis-Menten elimination kinetics].
Zhongguo Yao Li Xue Bao. 1986 Sep;7(5):385-9.
6
Nonlinear pharmacokinetics of ethanol elimination in long sleep and short sleep mice.
Alcohol Clin Exp Res. 1983 Winter;7(1):95-9. doi: 10.1111/j.1530-0277.1983.tb05420.x.
7
Michaelis-Menten elimination kinetics: areas under curves, steady-state concentrations, and clearances for compartment models with different types of input.米氏消除动力学:不同输入类型的房室模型的曲线下面积、稳态浓度和清除率
Biopharm Drug Dispos. 1985 Apr-Jun;6(2):177-200. doi: 10.1002/bdd.2510060209.
8
Properties of the Michaelis-Menten equation and its integrated form which are useful in pharmacokinetics.米氏方程及其积分形式在药代动力学中有用的性质。
J Pharmacokinet Biopharm. 1973 Apr;1(2):103-21. doi: 10.1007/BF01059625.
9
Michaelis-Menten metabolite formation kinetics: equations relating area under the curve and metabolite recovery to the administered dose.米氏代谢物形成动力学:将曲线下面积和代谢物回收率与给药剂量相关联的方程式。
J Pharm Sci. 1990 Oct;79(10):902-6. doi: 10.1002/jps.2600791012.
10
On the identification of Michaelis-Menten elimination parameters from a single dose-response curve.关于从单剂量反应曲线识别米氏消除参数
J Pharmacokinet Biopharm. 1984 Apr;12(2):193-221. doi: 10.1007/BF01059278.

引用本文的文献

1
Integrated equation to evaluate accumulation profiles of drugs eliminated by Michaelis-Menten kinetics.用于评估通过米氏动力学消除的药物蓄积曲线的综合方程。
J Pharmacokinet Biopharm. 1979 Apr;7(2):227-32. doi: 10.1007/BF01059740.
2
A tracer interaction method for nonlinear pharmacokinetics analysis: application to evaluation of nonlinear elimination.一种用于非线性药代动力学分析的示踪剂相互作用方法:在非线性消除评估中的应用。
J Pharmacokinet Biopharm. 1997 Oct;25(5):569-93. doi: 10.1023/a:1025765330455.
3
On the identification of Michaelis-Menten elimination parameters from a single dose-response curve.

本文引用的文献

1
Effects of solid food on blood levels of alcohol in man.固体食物对人体血液酒精水平的影响。
Res Commun Chem Pathol Pharmacol. 1976 Apr;13(4):713-22.
2
Blood ethanol concentrations during and following constant-rate intravenous infusion of alcohol.酒精恒速静脉输注期间及之后的血液乙醇浓度
Clin Pharmacol Ther. 1976 Feb;19(2):213-23. doi: 10.1002/cpt1976192213.
3
New method for detecting and quantitating pharmacokinetic drug-drug interactions applied to ethanol-propranolol.
关于从单剂量反应曲线识别米氏消除参数
J Pharmacokinet Biopharm. 1984 Apr;12(2):193-221. doi: 10.1007/BF01059278.
4
The deterministic identifiability of nonlinear pharmacokinetic models.非线性药代动力学模型的确定性可识别性
J Pharmacokinet Biopharm. 1984 Apr;12(2):177-91. doi: 10.1007/BF01059277.
Res Commun Chem Pathol Pharmacol. 1976 Jan;13(1):9-18.
4
Elimination of alcohol from human blood.人体血液中酒精的消除。
J Pharm Sci. 1976 Jan;65(1):152-4. doi: 10.1002/jps.2600650142.
5
Food effects on absorption and metabolism of alcohol.食物对酒精吸收和代谢的影响。
J Stud Alcohol. 1976 Sep;37(9):1197-214. doi: 10.15288/jsa.1976.37.1197.
6
Development of a dosage scheme for simultaneous intravenous and oral administration of mexiletine.
Postgrad Med J. 1977;53 Suppl 1:128-33.
7
Fasting and nonfasting blood ethanol concentrations following repeated oral administration of ethanol to one adult male subject.对一名成年男性受试者重复口服乙醇后空腹和非空腹血液中的乙醇浓度。
J Pharmacokinet Biopharm. 1977 Feb;5(1):41-52. doi: 10.1007/BF01064808.