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Biologically stable analogues of TRH with increased neuropharmacological potency.

作者信息

Brewster D, Dettmar P W, Metcalf G

出版信息

Neuropharmacology. 1981 May;20(5):497-503. doi: 10.1016/0028-3908(81)90184-2.

DOI:10.1016/0028-3908(81)90184-2
PMID:6787451
Abstract
摘要

相似文献

1
Biologically stable analogues of TRH with increased neuropharmacological potency.
Neuropharmacology. 1981 May;20(5):497-503. doi: 10.1016/0028-3908(81)90184-2.
2
Thyrotropin-releasing hormone (TRH) analogues show enhanced CNS selectivity because of increased biological stability.
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Behavioural and biochemical evidence for the release of noradrenaline in mouse brain by TRH and some of its biologically stable analogues.
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Neuropharmacological evaluation of RX 77368--a stabilised analogue of thyrotropin-releasing hormone (TRH).RX 77368的神经药理学评估——促甲状腺激素释放激素（TRH）的一种稳定类似物。
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Thermic and tremorogenic effects of thyroliberin (TRH) in reserpine-treated mice--the non-involvement of GABA-ergic mechanisms.促甲状腺素释放激素（TRH）对利血平处理小鼠的产热和致颤效应——γ-氨基丁酸能机制未参与其中
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The binding of 3H-(3-MeHis2) thyrotropin releasing hormone to brain membranes and temperature response to thyrotropin releasing hormone in different strains of mice.3H -（3 - 甲基组氨酸2）促甲状腺激素释放激素与不同品系小鼠脑膜的结合及对促甲状腺激素释放激素的温度反应
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Biochem Biophys Res Commun. 1982 Nov 30;109(2):556-61. doi: 10.1016/0006-291x(82)91757-0.

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Int J Nephrol Renovasc Dis. 2011;4:101-13. doi: 10.2147/IJNRD.S22783. Epub 2011 Jul 20.
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Antagonizing effects of YM-14673, a new TRH derivative, on behavioral and electroencephalographic changes in reserpinized animals.新型促甲状腺激素释放激素衍生物YM-14673对利血平化动物行为和脑电图变化的拮抗作用
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The effects of TRH analogues on cerebral ischaemia produced by middle cerebral artery occlusion in the rat.促甲状腺激素释放激素类似物对大鼠大脑中动脉闭塞所致脑缺血的影响。
Exp Brain Res. 1988;70(2):342-50. doi: 10.1007/BF00248359.
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Effects of a new TRH analogue, YM-14673 on the central nervous system.
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Electrophysiological observations in patients with motor neuron disease receiving a thyrotropin releasing hormone analogue (RX77368).接受促甲状腺激素释放激素类似物（RX77368）治疗的运动神经元病患者的电生理观察
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J Neurol Neurosurg Psychiatry. 1987 Oct;50(10):1359-70. doi: 10.1136/jnnp.50.10.1359.