新引入的β-内酰胺类抗生素对肾二肽酶的相对稳定性
Comparative stability of newly introduced beta-lactam antibiotics to renal dipeptidase.
作者信息
Mikami H, Ogashiwa M, Saino Y, Inoue M, Mitsuhashi S
出版信息
Antimicrob Agents Chemother. 1982 Oct;22(4):693-5. doi: 10.1128/AAC.22.4.693.
Abstract
Renal dipeptidase purified from swine kidney hydrolyzed N-formimidoyl thienamycin, carpetimycins A and B, and Sch29482, but not azthreonam, penicillin G, or cephaloridine.
摘要
从猪肾中纯化得到的肾二肽酶可水解N-甲脒基硫霉素、卡培霉素A和B以及Sch29482，但不能水解氨曲南、青霉素G或头孢菌素。
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本文引用的文献
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Protein measurement with the Folin phenol reagent.使用福林酚试剂进行蛋白质测定。
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Epithienamycins-novel beta-lactams related to thienamycin. I. Production and antibacterial activity.
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Carpetimycins A and B, new beta-lactam antibiotics.地毯霉素A和B，新型β-内酰胺抗生素。
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Azthreonam (SQ 26,776), a synthetic monobactam specifically active against aerobic gram-negative bacteria.氨曲南（SQ 26,776），一种对需氧革兰氏阴性菌有特效的合成单环β-内酰胺抗生素。
Antimicrob Agents Chemother. 1982 Jan;21(1):85-92. doi: 10.1128/AAC.21.1.85.
6
Effect of N-formimidoyl thienamycin (MK0787) on beta-lactamases and activity against beta-lactamase-producing strains.N-甲脒基硫霉素（MK0787）对β-内酰胺酶的作用及其对产β-内酰胺酶菌株的活性。
Antimicrob Agents Chemother. 1980 Nov;18(5):837-8. doi: 10.1128/AAC.18.5.837.
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8
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Thienamycin, a new beta-lactam antibiotic. I. Discovery, taxonomy, isolation and physical properties.硫霉素，一种新型β-内酰胺抗生素。I. 发现、分类学、分离及物理性质。
J Antibiot (Tokyo). 1979 Jan;32(1):1-12. doi: 10.7164/antibiotics.32.1.
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