通过用³H-阿扑吗啡和³H-多潘立酮进行结合研究鉴定出三类多巴胺受体（D-2、D-3、D-4）。 - Suppr

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Three classes of dopamine receptor (D-2, D-3, D-4) identified by binding studies with 3H-apomorphine and 3H-domperidone.

作者信息

Sokoloff P, Martres M P, Schwartz J C

出版信息

Naunyn Schmiedebergs Arch Pharmacol. 1980;315(2):89-102. doi: 10.1007/BF00499251.

DOI:10.1007/BF00499251

PMID:7207647

Abstract

摘要

相似文献

Three classes of dopamine receptor (D-2, D-3, D-4) identified by binding studies with 3H-apomorphine and 3H-domperidone.通过用³H-阿扑吗啡和³H-多潘立酮进行结合研究鉴定出三类多巴胺受体（D-2、D-3、D-4）。

Naunyn Schmiedebergs Arch Pharmacol. 1980;315(2):89-102. doi: 10.1007/BF00499251.

3H-apomorphine labels both dopamine postsynaptic receptors and autoreceptors.3H-阿扑吗啡标记多巴胺突触后受体和自身受体。

Nature. 1980 Nov 20;288(5788):283-6. doi: 10.1038/288283a0.

Dopamine receptors in the goldfish retina: 3H-spiroperidol and 3H-domperidone binding; and dopamine-stimulated adenylate cyclase activity.金鱼视网膜中的多巴胺受体：3H-螺哌啶醇和3H-多潘立酮结合；以及多巴胺刺激的腺苷酸环化酶活性。

Life Sci. 1980 Jul 7;27(1):23-31. doi: 10.1016/0024-3205(80)90015-6.

Guanine nucleotides distinguish between two dopamine receptors.鸟嘌呤核苷酸可区分两种多巴胺受体。

Nature. 1979 Apr 5;278(5704):577-8. doi: 10.1038/278577a0.

Kainate lesion dissociates striatal dopamine receptor radioligand binding sites.海人酸损伤使纹状体多巴胺受体放射性配体结合位点解离。

Eur J Pharmacol. 1981 Mar 5;70(1):71-5. doi: 10.1016/0014-2999(81)90434-9.

Characterization of 3H-domperidone binding on striatal dopamine receptors.3H-多潘立酮与纹状体多巴胺受体结合的特性研究。

Life Sci. 1978 Oct 30;23(17-18):1781-4. doi: 10.1016/0024-3205(78)90108-x.

The effects of (-)N-(chloroethyl)-norapomorphine on [3H]-apomorphine binding to striatal dopamine receptors.（-）N-（氯乙基）-去甲阿扑吗啡对[3H]-阿扑吗啡与纹状体多巴胺受体结合的影响。

Biochem Pharmacol. 1982 Nov 15;31(22):3693-4. doi: 10.1016/0006-2952(82)90599-8.

Effects of dopaminergic agonists and antagonists on [3H]apomorphine binding to striatal membranes: sulpiride lack of interactions with positive cooperative [3H]apomorphine binding.多巴胺能激动剂和拮抗剂对[3H]阿扑吗啡与纹状体膜结合的影响：舒必利与正协同[3H]阿扑吗啡结合缺乏相互作用。

Brain Res. 1980 Oct 20;199(2):335-42. doi: 10.1016/0006-8993(80)90693-9.

Selective labelling of dopamine (D2) receptors in rat striatum by [3H]domperidone but not by [3H]spiperone.[3H]多潘立酮可对大鼠纹状体中的多巴胺（D2）受体进行选择性标记，而[3H]螺哌隆则不能。

Eur J Pharmacol. 1982 Jul 9;81(2):273-85. doi: 10.1016/0014-2999(82)90445-9.

Quantitative determination of dopamine receptor subtypes not linked to activation of adenylate cyclase in rat striatum.大鼠纹状体中与腺苷酸环化酶激活无关的多巴胺受体亚型的定量测定。

Proc Natl Acad Sci U S A. 1982 Dec;79(23):7561-5. doi: 10.1073/pnas.79.23.7561.

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Chronic molindone treatment: relative inability to elicit dopamine receptor supersensitivity in rats.慢性吗茚酮治疗：大鼠中相对无法引发多巴胺受体超敏反应

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Dopaminergic binding sites in rat striatal slices and the action of guanyl nucleotides.大鼠纹状体切片中的多巴胺能结合位点及鸟苷酸的作用。

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3H-Dopamine binding sites differ in rat striatum and pituitary.3H-多巴胺结合位点在大鼠纹状体和垂体中存在差异。

Naunyn Schmiedebergs Arch Pharmacol. 1984 Sep;327(3):221-7. doi: 10.1007/BF00502453.

Differential anatomical location of [3H]-N,n-propylnorapomorphine and [3H]-spiperone binding sites in the striatum and substantia nigra of the rat.大鼠纹状体和黑质中[3H]-N，N-丙基去甲阿朴吗啡和[3H]-螺哌隆结合位点的差异解剖位置。

Br J Pharmacol. 1983 Jun;79(2):599-610. doi: 10.1111/j.1476-5381.1983.tb11035.x.

Sodium ion modulates D2 receptor characteristics of dopamine agonist and antagonist binding sites in striatum and retina.钠离子调节纹状体和视网膜中多巴胺激动剂和拮抗剂结合位点的D2受体特性。

Proc Natl Acad Sci U S A. 1982 Jul;79(13):4212-6. doi: 10.1073/pnas.79.13.4212.

本文引用的文献

Protein measurement with the Folin phenol reagent.使用福林酚试剂进行蛋白质测定。

J Biol Chem. 1951 Nov;193(1):265-75.

3H-apomorphine labels both dopamine postsynaptic receptors and autoreceptors.3H-阿扑吗啡标记多巴胺突触后受体和自身受体。

Nature. 1980 Nov 20;288(5788):283-6. doi: 10.1038/288283a0.

Effect of kainic acid on striatal dopamine receptors.海人酸对纹状体多巴胺受体的影响。

Brain Res. 1980 Oct 6;198(2):491-6. doi: 10.1016/0006-8993(80)90766-0.

Quantitative assessment of heterogeneous 3H-spiperone binding to rat neostriatum and frontal cortex.对大鼠新纹状体和额叶皮质中异质性3H-螺哌隆结合的定量评估。

Life Sci. 1980 Feb 18;26(7):511-7. doi: 10.1016/0024-3205(80)90313-6.

Endogenous components of the striatum confer dopamine-sensitivity upon adenylate cyclase activity: the role of endogenous guanyl nucleotides.纹状体的内源性成分赋予腺苷酸 cyclase 活性多巴胺敏感性：内源性鸟苷酸的作用。

Brain Res. 1980 Jan 6;181(1):139-49. doi: 10.1016/0006-8993(80)91264-0.

The role of hormone receptors and GTP-regulatory proteins in membrane transduction.激素受体和GTP调节蛋白在膜转导中的作用。

Nature. 1980 Mar 6;284(5751):17-22. doi: 10.1038/284017a0.

Pharmacological estimation of drug-receptor dissociation constants. Statistical evaluation. I. Agonists.药物-受体解离常数的药理学估算。统计学评估。I. 激动剂。

J Pharmacol Exp Ther. 1971 Apr;177(1):1-12.

Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction.抑制常数（K1）与导致酶促反应50%抑制率（I50）的抑制剂浓度之间的关系。

Biochem Pharmacol. 1973 Dec 1;22(23):3099-108. doi: 10.1016/0006-2952(73)90196-2.

Antagonistic effects of apomorphine and haloperidol on rat striatal synaptosomal tyrosine hydroxylase.阿扑吗啡和氟哌啶醇对大鼠纹状体突触体酪氨酸羟化酶的拮抗作用。

J Pharm Pharmacol. 1974 May;26(5):367-9. doi: 10.1111/j.2042-7158.1974.tb09293.x.

Drug-induced changes in the release of 3 H-monoamines from field stimulated rat brain slices.药物诱导的大鼠脑片经场刺激后3H-单胺释放的变化。

Acta Physiol Scand Suppl. 1971;371:35-44. doi: 10.1111/j.1748-1716.1971.tb05213.x.

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