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利培酮过量。

Overdose of risperidone.

作者信息

Brown K, Levy H, Brenner C, Leffler S, Hamburg E L

机构信息

Division of Emergency Medicine, University of New Mexico Medical Center, Albuquerque.

出版信息

Ann Emerg Med. 1993 Dec;22(12):1908-10. doi: 10.1016/s0196-0644(05)80421-4.

DOI:10.1016/s0196-0644(05)80421-4
PMID:7694530
Abstract

Risperidone is an investigational antipsychotic agent currently being tested in an international multicenter drug trial. We report the first case of a risperidone overdose in an apparent suicide attempt. This was without serious clinical side effects and manifested mainly as ECG abnormalities.

摘要

利培酮是一种正在国际多中心药物试验中进行测试的研究性抗精神病药物。我们报告了首例因明显自杀企图而过量服用利培酮的病例。该病例无严重临床副作用,主要表现为心电图异常。

相似文献

1
Overdose of risperidone.利培酮过量。
Ann Emerg Med. 1993 Dec;22(12):1908-10. doi: 10.1016/s0196-0644(05)80421-4.
2
Paliperidone overdose with delayed onset of toxicity.帕利哌酮过量致迟发性中毒。
Ann Emerg Med. 2011 Jul;58(1):80-2. doi: 10.1016/j.annemergmed.2010.10.015. Epub 2011 Mar 4.
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New antipsychotic agent, risperidone, introduced.
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Risperidone: the search for a better antipsychotic.利培酮:寻找更好的抗精神病药物。
Perspect Psychiatr Care. 1995 Jan-Mar;31(1):30-3. doi: 10.1111/j.1744-6163.1995.tb00455.x.
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New clinical manifestations of acute risperidone poisoning.急性利培酮中毒的新临床表现。
J Toxicol Clin Toxicol. 1999;37(7):893-5. doi: 10.1081/clt-100102531.
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A case of risperidone overdose in early schizophrenia: a review of potential complications.一例早期精神分裂症患者利培酮过量:潜在并发症综述
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Effects of risperidone on motor and sexual activity in the rat.
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FDA approved new drug bulletin: risperidone (risperdal).美国食品药品监督管理局批准的新药公告:利培酮(维思通)。
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引用本文的文献

1
Inhibition of cloned hERG potassium channels by risperidone and paliperidone.利培酮和帕利哌酮对克隆的人乙醚 - 去极化激活钾通道(hERG)的抑制作用
Naunyn Schmiedebergs Arch Pharmacol. 2017 Jun;390(6):633-642. doi: 10.1007/s00210-017-1364-5. Epub 2017 Mar 6.
2
QTc interval prolongation and torsade de pointes associated with second-generation antipsychotics and antidepressants: a comprehensive review.第二代抗精神病药和抗抑郁药相关的QTc间期延长及尖端扭转型室性心动过速:一项综述
CNS Drugs. 2014 Oct;28(10):887-920. doi: 10.1007/s40263-014-0196-9.
3
Risperidone, QTc interval prolongation, and torsade de pointes: a systematic review of case reports.
利培酮、QTc 间期延长和尖端扭转型室性心动过速:病例报告的系统评价。
Psychopharmacology (Berl). 2013 Aug;228(4):515-24. doi: 10.1007/s00213-013-3192-8. Epub 2013 Jun 30.
4
Antipsychotic-induced hyponatraemia: a systematic review of the published evidence.抗精神病药引起的低钠血症:已发表证据的系统评价。
Drug Saf. 2010 Feb 1;33(2):101-14. doi: 10.2165/11319070-000000000-00000.
5
A systematic review of cardiovascular effects after atypical antipsychotic medication overdose.非典型抗精神病药物过量后心血管效应的系统评价。
Am J Emerg Med. 2009 Jun;27(5):607-16. doi: 10.1016/j.ajem.2008.04.020.
6
Risperidone-induced action potential prolongation is attenuated by increased repolarization reserve due to concomitant block of I(Ca,L).由于同时阻断L型钙电流(I(Ca,L))使复极储备增加,从而减轻了利培酮诱导的动作电位延长。
Naunyn Schmiedebergs Arch Pharmacol. 2005 May;371(5):393-400. doi: 10.1007/s00210-005-1063-5. Epub 2005 Jun 16.
7
Atypical antipsychotics: from potassium channels to torsade de pointes and sudden death.非典型抗精神病药物:从钾通道到尖端扭转型室速和猝死
Drug Saf. 2005;28(1):35-51. doi: 10.2165/00002018-200528010-00003.
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New Generation Antipsychotic Drugs and QTc Interval Prolongation.新一代抗精神病药物与QTc间期延长
Prim Care Companion J Clin Psychiatry. 2003 Oct;5(5):205-215. doi: 10.4088/pcc.v05n0504.
9
A risk-benefit assessment of risperidone in schizophrenia.利培酮治疗精神分裂症的风险效益评估。
Drug Saf. 1995 Feb;12(2):139-45. doi: 10.2165/00002018-199512020-00006.
10
Risperidone. A review of its pharmacology and therapeutic potential in the treatment of schizophrenia.利培酮。其药理学及治疗精神分裂症的潜在疗效综述。
Drugs. 1994 Aug;48(2):253-73. doi: 10.2165/00003495-199448020-00009.