新型3,5-二氨基异噻唑衍生物的合成及其抗菌活性
Synthesis and antimicrobial activity of new 3,5-diaminoisothiazole derivatives.
作者信息
Cocco M T, Congiu C, Maccioni A, Onnis V, Schivo M L, De Logu A
出版信息
Farmaco. 1994 Feb;49(2):137-40.
PMID:8003183
Abstract
The 3,5-diaminoisothiazole derivatives 23-42 were synthesized in excellent yields by oxidative cyclization of 3-amino-3-(dialkylamino)propenethioamide derivatives. These intermediates and the isothiazole derivatives were tested in vitro for their antimicrobial activity.
摘要
通过3-氨基-3-(二烷基氨基)丙烯硫酰胺衍生物的氧化环化反应，以优异的产率合成了3,5-二氨基异噻唑衍生物23 - 42。对这些中间体和异噻唑衍生物进行了体外抗菌活性测试。
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