Adenosine A1 receptor agonists as clinically viable agents for treatment of ischemic brain disorders.
作者信息
Bischofberger N, Jacobson K A, von Lubitz D K
机构信息
Gilead Sciences, Inc., Foster City, California 94404, USA.
出版信息
Ann N Y Acad Sci. 1997 Oct 15;825:23-9. doi: 10.1111/j.1749-6632.1997.tb48411.x.
Abstract
摘要
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本文引用的文献
1
Species Differences in Ligand Affinity at Central A-Adenosine Receptors.中枢A1-腺苷受体配体亲和力的种属差异。
Drug Dev Res. 1994 Sep;33(1):51-59. doi: 10.1002/ddr.430330109.
2
N-substituted adenosines as novel neuroprotective A(1) agonists with diminished hypotensive effects.
J Med Chem. 1999 Sep 9;42(18):3463-77. doi: 10.1021/jm960682u.
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Postischemic administration of adenosine amine congener (ADAC): analysis of recovery in gerbils.腺苷胺类似物（ADAC）缺血后给药：沙土鼠恢复情况分析
Eur J Pharmacol. 1996 Dec 5;316(2-3):171-9. doi: 10.1016/s0014-2999(96)00667-x.
4
Adenosine receptor ligands: differences with acute versus chronic treatment.腺苷受体配体：急性治疗与慢性治疗的差异
Trends Pharmacol Sci. 1996 Mar;17(3):108-13. doi: 10.1016/0165-6147(96)10002-x.
5
Reduction of postischemic brain damage and memory deficits following treatment with the selective adenosine A1 receptor agonist.使用选择性腺苷A1受体激动剂治疗后，缺血性脑损伤和记忆缺陷减轻。
Eur J Pharmacol. 1996 Apr 29;302(1-3):43-8. doi: 10.1016/0014-2999(96)00101-x.
6
The A3 adenosine receptor is the unique adenosine receptor which facilitates release of allergic mediators in mast cells.A3 腺苷受体是唯一能促进肥大细胞释放过敏介质的腺苷受体。
J Biol Chem. 1993 Aug 15;268(23):16887-90.
7
Chronic administration of selective adenosine A1 receptor agonist or antagonist in cerebral ischemia.在脑缺血中选择性腺苷A1受体激动剂或拮抗剂的长期给药。
Eur J Pharmacol. 1994 Apr 21;256(2):161-7. doi: 10.1016/0014-2999(94)90241-0.
8
Chronic adenosine A1 receptor agonist and antagonist: effect on receptor density and N-methyl-D-aspartate induced seizures in mice.慢性腺苷A1受体激动剂和拮抗剂：对小鼠受体密度及N-甲基-D-天冬氨酸诱导癫痫发作的影响
Eur J Pharmacol. 1994 Feb 21;253(1-2):95-9. doi: 10.1016/0014-2999(94)90762-5.
9
Adenosine: a prototherapeutic concept in neurodegeneration.腺苷：神经退行性变中的一种原治疗概念。
Ann N Y Acad Sci. 1995 Sep 15;765:163-78; discussion 196-7. doi: 10.1111/j.1749-6632.1995.tb16573.x.
10
Endogenously released adenosine regulates excitability in the in vitro hippocampus.内源性释放的腺苷调节体外培养海马体的兴奋性。
Epilepsia. 1980 Oct;21(5):541-8. doi: 10.1111/j.1528-1157.1980.tb04305.x.
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