Ahmed M, Shikha H A, Sadhu S K, Rahman M T, Datta B K
Department of Pharmacy, University of Dhaka, Dhaka, Bangladesh.
Pharmazie. 2001 Aug;56(8):657-60.
Scoparinol, a diterpene, isolated from Scoparia dulcis showed significant analgesic (p < 0.001) and anti-inflammatory activity (p < 0.01) in animals. A sedative action of scoparinol was demonstrated by a marked potentiation of pentobarbital-induced sedation with a significant effect on both onset and duration of sleep (p < 0.05). Measurement of urine volume after administration of scoparinol indicated its significant diuretic action.
从甜地丁中分离得到的二萜类化合物scoparinol在动物实验中显示出显著的镇痛作用(p < 0.001)和抗炎活性(p < 0.01)。scoparinol对戊巴比妥诱导的镇静有明显的增强作用,对睡眠的起始和持续时间均有显著影响(p < 0.05),表明其具有镇静作用。scoparinol给药后尿量的测量表明其具有显著的利尿作用。